Target Details
| UniProt AC | Q9NSY1 |
|---|---|
| Gene Symbol | BMP2K |
| Protein Name | BMP-2-inducible protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15282 (BMP2K_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 111
- Clinical molecules 18
- Avg pChEMBL 7.15
KEGG Pathways (1)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLGZSRKKPYFWHZ
|
9.7 | Kd | 6 | — | |
ZCCPLJOKGAACRT
|
8.9 | Kd | 599 | — | |
XZXHXSATPCNXJR
|
8.7 | Kd | 165 | Yes | |
NEQZWEXWOFPKOT
|
8.4 | Kd | 9 | — | |
WINHZLLDWRZWRT
|
8.3 | Kd | 201 | Yes | |
HKSZLNNOFSGOKW
|
8.2 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
8.2 | Kd | 213 | — | |
PFMMJDPMFCVRCB
|
8.2 | IC50 | 4 | — | |
YFNWWNRZJGMDBR
|
8.2 | Kd | 35 | — | |
RSFALMGMTQBFJZ
|
8.1 | Kd | 9 | — | |
XLSYZSRXVVCHLS
|
8.1 | Kd | 48 | — | |
YYLKKYCXAOBSRM
|
8.0 | Kd | 191 | — | |
FFTUIKFDUYMWTI
|
8.0 | IC50 | 5 | — | |
HJDMEPOCEJXNJU
|
7.9 | Ki | 3 | — | |
IPEXHQGMTHOKQV
|
7.9 | Kd | 12 | — | |
ALKJNCZNEOTEMP
|
7.8 | Kd | 55 | — | |
RYYNGWLOYLRZLK
|
7.8 | Kd | 45 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
SENOTLIGBLGKGP
|
7.8 | Ki | 3 | — | |
UCBIQZUJJSVQHL
|
7.8 | Ki | 8 | — | |
USXZHEGWWNBLBI
|
7.8 | Ki | 4 | — | |
GXQWWDBZTZLIAJ
|
7.7 | Ki | 3 | — | |
OSVUGUHRKMMBSE
|
7.7 | Kd | 170 | — | |
NKCMEGZSWOVKIL
|
7.7 | Ki | 3 | — | |
SVNVPNHWFJFRLZ
|
7.7 | IC50 | 8 | — | |
XUZMWHLSFXCVMG
|
7.7 | Kd | 24 | — | |
NXSJMRCTGYTSTK
|
7.6 | Kd | 200 | — | |
IBPRZGYJJMUZLP
|
7.6 | IC50 | 2 | — | |
JKCNRFQYOHWEDM
|
7.6 | IC50 | 2 | — | |
KRIUNPBAQZGFQA
|
7.6 | Kd | 76 | — | |
NSQIWTMRSLRZLP
|
7.6 | IC50 | 2 | — | |
OVUOFYVATYZDTQ
|
7.6 | IC50 | 2 | — | |
RJNDAWMSDOWAKQ
|
7.6 | IC50 | 2 | — | |
ZZVWLSVVRDNANL
|
7.6 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.6 | Kd | 151 | — | |
NTOMZGNNDKIPEH
|
7.6 | Ki | 4 | — | |
JEESDCKVMQTTMP
|
7.5 | Ki | 3 | — | |
ZVSNSFQQKSZZMY
|
7.5 | IC50 | 7 | — | |
JOOXLOJCABQBSG
|
7.5 | Kd | 139 | — | |
CJIAUJUVHMAHQC
|
7.5 | Ki | 4 | — | |
GOOYSJIWTIHOGW
|
7.5 | IC50 | 3 | — | |
LOLPPWBBNUVNQZ
|
7.5 | Kd | 97 | Yes | |
YSMDVXCUNQWGNN
|
7.4 | Ki | 4 | — | |
DPCPNRYPXUUJCP
|
7.4 | Ki | 4 | — | |
RDROKTFULACVDQ
|
7.4 | IC50 | 8 | — | |
HWXVIOGONBBTBY
|
7.4 | Kd | 27 | — | |
OEZHSZIDGUKBRK
|
7.4 | IC50 | 10 | — | |
MCYCSSJHDPRHBZ
|
7.4 | Ki | 4 | — | |
OYONTEXKYJZFHA
|
7.3 | Kd | 69 | Yes | |
JNYMSOJGKCXZLV
|
7.3 | Ki | 3 | — |