Target Details
| UniProt AC | Q9NS75 |
|---|---|
| Gene Symbol | CYSLTR2 |
| Protein Name | Cysteinyl leukotriene receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 378
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (378)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LUCQNYBUJLHCPS
|
10.5 | IC50 | 2 | — | |
SDTNBOHERRYJEY
|
10.2 | IC50 | 2 | — | |
YSEIYPQSNRDRHK
|
10.0 | Ki | 2 | — | |
CSIBKBIBULLMDV
|
10.0 | IC50 | 2 | — | |
VOENOFDVFYQPAQ
|
9.8 | IC50 | 2 | — | |
PITFCUBRHKJFAT
|
9.8 | IC50 | 2 | — | |
ZWMCRMIDWSXPOI
|
9.8 | IC50 | 2 | — | |
AXUZQJFHDNNPFG
|
9.7 | Ki | 2 | — | |
BFNAFTJCDGWFMQ
|
9.7 | IC50 | 2 | — | |
ZYFXZSJLWGWRDB
|
9.7 | Ki | 2 | — | |
DPIZIIGHFHBBGL
|
9.6 | Ki | 2 | — | |
SKOXHEZNXXKBOY
|
9.6 | Ki | 2 | — | |
AILQNBFWBWZOJI
|
9.5 | Ki | 2 | — | |
GOUWWDPQGZJWEW
|
9.5 | Ki | 2 | — | |
HOTVSPQKJFKWJW
|
9.5 | Ki | 2 | — | |
LJGSYVAEVXDQCR
|
9.5 | Ki | 2 | — | |
OHCBAIWHQUWKQY
|
9.5 | Ki | 2 | — | |
RHXDSNDNDGKMLP
|
9.5 | IC50 | 2 | — | |
WRGRFTHOWDHZCX
|
9.5 | Ki | 2 | — | |
KQXMBUWEISAGDL
|
9.5 | IC50 | 2 | — | |
KEGQUGIJAFPXHO
|
9.5 | IC50 | 2 | — | |
BRYNGLQFTGZDFD
|
9.5 | IC50 | 2 | — | |
KDIPHOWDGBZABT
|
9.5 | IC50 | 2 | — | |
OSSGVJHRBLHMLQ
|
9.4 | IC50 | 2 | — | |
CILFBYXDVWMEGJ
|
9.4 | IC50 | 2 | — | |
QCBBZDIVKHHUTB
|
9.4 | IC50 | 2 | — | |
OQPSKUCABGKHFR
|
9.4 | IC50 | 2 | — | |
MHHBMEJREHQZQU
|
9.4 | IC50 | 2 | — | |
YRCPIXCRSAKRGM
|
9.3 | IC50 | 2 | — | |
YEFODJIFJVHEIS
|
9.3 | IC50 | 2 | — | |
QZECKERBZPCVOV
|
9.3 | IC50 | 2 | — | |
ODBOCKWNRNDVQH
|
9.3 | IC50 | 2 | — | |
AFIGUFVMDMNGJX
|
9.3 | Ki | 2 | — | |
DGUXLXDTCHULNE
|
9.3 | IC50 | 2 | — | |
JHKPLZCCMOGUEI
|
9.3 | IC50 | 2 | — | |
YTYZMTWLPBHKJN
|
9.3 | IC50 | 2 | — | |
UCHDWCPVSPXUMX
|
9.3 | IC50 | 6 | — | |
CKLRKPMEGUXCIX
|
9.3 | IC50 | 2 | — | |
SOUXTOZGVBFBFE
|
9.3 | IC50 | 2 | — | |
DUCNKECWDRIBHL
|
9.2 | IC50 | 2 | — | |
APMBFPQCZFCKCO
|
9.2 | IC50 | 2 | — | |
LITAULXAAATXRV
|
9.2 | IC50 | 2 | — | |
BYTUMFJCBKNJKZ
|
9.2 | IC50 | 2 | — | |
IGUFQFBMEPZVOT
|
9.2 | IC50 | 2 | — | |
IISZUJHNGQJOEV
|
9.2 | IC50 | 2 | — | |
PNHUIGYHBQXQAN
|
9.2 | IC50 | 2 | — | |
JQQVCFPPEBPPIO
|
9.2 | IC50 | 2 | — | |
LRXDBHMSRBIJLN
|
9.2 | Ki | 2 | — | |
IOGVHXVJWAEZRZ
|
9.1 | IC50 | 2 | — | |
NBQKINXMPLXUET
|
9.1 | IC50 | 2 | — |