Target Details
| UniProt AC | Q9NRM7 |
|---|---|
| Gene Symbol | LATS2 |
| Protein Name | Serine/threonine-protein kinase LATS2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 84
- Clinical molecules 6
- Avg pChEMBL 7.33
KEGG Pathways (3)
Active Molecules (84)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXRCZLGBPPMVSP
|
6.6 | Kd | 9 | — | |
UFYSVZDHPHLSEY
|
6.5 | IC50 | 2 | — | |
FFSAICURRWPYFX
|
6.4 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
PTPZOJYJIOCLLO
|
6.4 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
RJTQBPCQZQSZFF
|
6.3 | Kd | 9 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
CHYCCNFSSCTALZ
|
6.3 | IC50 | 2 | — | |
IZKUFWOXLYUAAV
|
6.3 | IC50 | 2 | — | |
CCJRVCDZHWNBTA
|
6.3 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
KPAQBWXRTMKVCB
|
6.2 | IC50 | 2 | — | |
GMBDJMAWOMXCHX
|
6.2 | IC50 | 2 | — | |
CELWQJHESXUCFF
|
6.2 | IC50 | 2 | — | |
WIFZIPRZHKCGGL
|
6.2 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
ZCBUQCWBWNUWSU
|
6.2 | Kd | 59 | — | |
ATBSEYKJNNUJPS
|
6.2 | IC50 | 2 | — | |
RKAHOQATMSONTM
|
6.2 | IC50 | 6 | — | |
UCTAUHCKGLOZHU
|
6.2 | IC50 | 2 | — | |
LFAHWMOZPVCJAY
|
6.1 | Kd | 8 | — | |
LMLFNPDYWJFFPD
|
6.1 | IC50 | 2 | — | |
VXYPJGHKVFBNME
|
6.1 | IC50 | 2 | — | |
WIFZIPRZHKCGGL
|
6.1 | IC50 | 2 | — | |
MBMKHDKGWLLWJM
|
6.1 | IC50 | 2 | — | |
BEZHNWWMIVIPFV
|
6.0 | IC50 | 2 | — | |
MGSXOJRYNIPSTE
|
6.0 | IC50 | 2 | — | |
QLNKJSSYMWYESY
|
6.0 | IC50 | 2 | — | |
GSFWSEGLHKYRGG
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MYPGOQOVEQKGDN
|
6.0 | IC50 | 2 | — |