Target Details
| UniProt AC | Q9NRM7 |
|---|---|
| Gene Symbol | LATS2 |
| Protein Name | Serine/threonine-protein kinase LATS2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 84
- Clinical molecules 6
- Avg pChEMBL 7.33
KEGG Pathways (3)
Active Molecules (84)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UAPFATLGRSUIKX
|
10.2 | Ki | 2 | — | |
SYHRTOREQDHSNY
|
10.2 | Ki | 2 | — | |
SAQSMANEGRAMNT
|
10.1 | Ki | 2 | — | |
SAQSMANEGRAMNT
|
10.1 | Ki | 2 | — | |
WEAHURJZQJBTGH
|
10.1 | Ki | 2 | — | |
JQAXPHDIJOQPBP
|
10.1 | Ki | 2 | — | |
DTVNECWMYCSEBL
|
9.9 | Ki | 2 | — | |
DTVNECWMYCSEBL
|
9.9 | Ki | 2 | — | |
PANBXEPRTUWMHA
|
9.4 | Ki | 2 | — | |
SXOIZZVBAAACIQ
|
9.0 | Ki | 2 | — | |
PTTKHXBEPPAXSE
|
9.0 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
9.0 | Kd | 289 | Yes | |
RGIKJUZEMMTILQ
|
8.7 | IC50 | 2 | — | |
SBPQHDLJGZBWTL
|
8.7 | IC50 | 2 | — | |
AFJHACZNTJKCIF
|
8.4 | IC50 | 2 | — | |
HQFDCITUHVQXEV
|
8.4 | IC50 | 2 | — | |
OLUIHIBCEWNDET
|
8.4 | IC50 | 2 | — | |
SBPQHDLJGZBWTL
|
8.2 | IC50 | 2 | — | |
JDMAQIORUXZAGZ
|
8.1 | IC50 | 2 | — | |
NCWUWMQIMGPXQR
|
8.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.1 | IC50 | 408 | — | |
DCIPFXLSLUFVQA
|
8.0 | IC50 | 2 | — | |
JVCDXTHYVYGMQC
|
7.9 | IC50 | 2 | — | |
GTDNROOVOBKLDL
|
7.8 | IC50 | 2 | — | |
TWSFYAXEDIOFFN
|
7.8 | IC50 | 2 | — | |
HVEXJKQESNIDLM
|
7.8 | Kd | 10 | — | |
SBPQHDLJGZBWTL
|
7.8 | IC50 | 2 | — | |
OJKBHNAVTDJSIO
|
7.7 | IC50 | 2 | — | |
GPKFECYSQTWZCI
|
7.7 | IC50 | 2 | — | |
RQCQSMAAAMSVHQ
|
7.7 | IC50 | 2 | — | |
IDYBIWQRAAGTKU
|
7.6 | IC50 | 2 | — | |
OCRGFIAWWYJUTP
|
7.5 | IC50 | 2 | — | |
RQXXATOWBUCCAY
|
7.5 | IC50 | 2 | — | |
WNBNLESOAUCHBN
|
7.5 | IC50 | 2 | — | |
VWCSZVWZRTZNCH
|
7.4 | Kd | 8 | — | |
WKYHVIILYCJVBF
|
7.3 | IC50 | 2 | — | |
ZFZNIZVNKXAOHL
|
7.3 | IC50 | 2 | — | |
RAXZSEGXMBWYQK
|
7.3 | Kd | 21 | — | |
ACTDLFQRJKPKFQ
|
7.2 | IC50 | 2 | — | |
PGOCRNZIASOKRK
|
7.2 | IC50 | 2 | — | |
IEDDDZFQZKDRBJ
|
7.2 | IC50 | 9 | — | |
KCWQIAOSJJWFIG
|
7.0 | IC50 | 2 | — | |
VCWNZJZLJJLTBZ
|
6.9 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.9 | Kd | 200 | — | |
KGPGFQWBCSZGEL
|
6.8 | Kd | 59 | Yes | |
YXFRTVUVQNPAHF
|
6.8 | IC50 | 2 | — | |
JJNZJRXOAFOQOK
|
6.8 | IC50 | 2 | — | |
VJFDDNKVWALCBK
|
6.8 | IC50 | 2 | — | |
IKOCQBSJIXAKFW
|
6.7 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
6.7 | Kd | 170 | — |