Target Details
| UniProt AC | Q9NR22 |
|---|---|
| Gene Symbol | PRMT8 |
| Protein Name | Protein arginine N-methyltransferase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF06325 (PrmA) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 35
- Clinical molecules 0
- Avg pChEMBL 7.43
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XCZUYGFLWBJNCB
|
9.0 | IC50 | 4 | — | |
QVFVESAOLFEXQX
|
8.7 | IC50 | 3 | — | |
SPEGERVLTUWZPA
|
8.7 | IC50 | 5 | — | |
FMTVWAGUJRUAKE
|
8.4 | IC50 | 5 | — | |
LUBCTIQAZDQPJR
|
8.3 | IC50 | 5 | — | |
BOGKHDNBFDMRMG
|
8.2 | IC50 | 3 | — | |
KJHBJSSYYMWKLQ
|
8.0 | IC50 | 3 | — | |
PMGPJYJFQITHHT
|
8.0 | IC50 | 3 | — | |
TXSFQHHRYLAEMB
|
8.0 | IC50 | 3 | — | |
LIENDGUHQUTLMD
|
7.8 | IC50 | 3 | — | |
GJDVMSRIXJKBKJ
|
7.7 | IC50 | 3 | — | |
HHJFNFLLPHTDTH
|
7.7 | IC50 | 3 | — | |
QCPRDFJGTLMBCJ
|
7.7 | IC50 | 3 | — | |
CNSBKLBZNFFFRD
|
7.6 | IC50 | 3 | — | |
CNMWTZSRTFSQJJ
|
7.6 | IC50 | 5 | — | |
VZDPLMKEFMWBMM
|
7.6 | IC50 | 5 | — | |
AHBGFVBNHAXGOD
|
7.5 | IC50 | 3 | — | |
MOPCOJLFDMFKCS
|
7.5 | IC50 | 4 | — | |
DVZZYZNFLHFCPI
|
7.5 | IC50 | 7 | — | |
FYZDIUPNFFHKJM
|
7.4 | IC50 | 2 | — | |
MDBHVKTYIGBDLO
|
7.3 | IC50 | 3 | — | |
LIVCXRSDQOQURR
|
7.2 | IC50 | 3 | — | |
WJJPSVIYQWOSFK
|
7.2 | IC50 | 3 | — | |
YOCSLRCPVKLWMS
|
7.2 | IC50 | 3 | — | |
UMKLFWMQTDMELK
|
7.1 | IC50 | 5 | — | |
HVDMIAFOVVMNJF
|
7.0 | IC50 | 4 | — | |
ZXTYIIDDTFQCGV
|
6.9 | IC50 | 3 | — | |
UOYRGGRFVPHLEJ
|
6.8 | IC50 | 3 | — | |
HOTVGBQTCMXBLC
|
6.7 | IC50 | 3 | — | |
QMDKVNSQXPVCRD
|
6.7 | IC50 | 3 | — | |
KWRBLASCKRNYTH
|
6.5 | IC50 | 3 | — | |
VMIKTYCHSCYQBD
|
6.5 | IC50 | 3 | — | |
CJZMDZQZJNDMPE
|
6.3 | IC50 | 3 | — | |
OLFLGFYCUQONAR
|
6.2 | IC50 | 3 | — | |
DVIUIRPCVXVFSX
|
6.0 | IC50 | 3 | — |