Target Details
| UniProt AC | Q9NR21 |
|---|---|
| Gene Symbol | PARP11 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF02825 (WWE) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 6.78
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MPXAEYSGFKRDQM
|
7.2 | IC50 | 7 | — | |
RMIJZTKTCJJVSA
|
7.0 | IC50 | 4 | — | |
HWGQMRYQVZSGDQ
|
6.8 | IC50 | 7 | — | |
ANAUZAZPUGQDNM
|
6.7 | IC50 | 3 | — | |
FSNNMBVVDWKKCB
|
6.6 | IC50 | 6 | — | |
ZKXNKMALIYTLJE
|
6.3 | IC50 | 4 | — |