Target Details
| UniProt AC | Q9NR20 |
|---|---|
| Gene Symbol | DYRK4 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 139
- Clinical molecules 1
- Avg pChEMBL 6.45
Active Molecules (139)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JBWDTSLHUJHODF
|
6.2 | IC50 | 9 | — | |
USYASDQVUTWEQM
|
6.2 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
6.2 | IC50 | 9 | — | |
CBTNARFZVOPLBO
|
6.2 | IC50 | 8 | — | |
HGMCNIGKEVZHFM
|
6.2 | IC50 | 8 | — | |
URXJBXVGNBGIJA
|
6.2 | IC50 | 9 | — | |
IJFKKIMDRSZOOW
|
6.1 | IC50 | 8 | — | |
PEICIAVUWSXRGP
|
6.1 | IC50 | 7 | — | |
XCTYEZWILVGTGO
|
6.1 | IC50 | 9 | — | |
XTJRKTBELWGSDN
|
6.1 | IC50 | 6 | — | |
HJEKFRDOAYXXRU
|
6.1 | IC50 | 8 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
FSWFKKQQSQHIRZ
|
6.1 | Ki | 10 | — | |
LRZYYIZFBXFSJB
|
6.1 | Ki | 69 | — | |
OEVQTWCGWDOIFZ
|
6.1 | IC50 | 7 | — | |
RLTCEYSNDOXWKS
|
6.1 | IC50 | 9 | — | |
RUQXGVGYNKIGJD
|
6.1 | IC50 | 9 | — | |
GHQYHWMWJLSKRP
|
6.1 | IC50 | 9 | — | |
WFOMWAYINPJPDX
|
6.1 | IC50 | 9 | — | |
XXIXFZAUCITSCM
|
6.1 | IC50 | 7 | — | |
GCSZJMUFYOAHFY
|
6.0 | IC50 | 8 | — | |
JBWDTSLHUJHODF
|
6.0 | IC50 | 8 | — | |
RYWACTNAXCMTTN
|
6.0 | IC50 | 9 | — | |
FIVWKNZKXNNFCW
|
6.0 | IC50 | 9 | — | |
FRPGBGWSLAGPND
|
6.0 | IC50 | 7 | — | |
LZTDWHFXSWDVAG
|
6.0 | IC50 | 7 | — | |
ROPFCXUWNMYMSW
|
6.0 | IC50 | 10 | — | |
AMBKAVGTUWUVBS
|
6.0 | IC50 | 8 | — | |
YYSXUOHHBBMQMJ
|
6.0 | IC50 | 7 | — | |
BDMXFIMYKGLQAL
|
6.0 | IC50 | 9 | — | |
AOBLBPWPSKBHSI
|
6.0 | Ki | 55 | — | |
BBCSUMURJUYILA
|
6.0 | IC50 | 9 | — | |
CHTMRWQLNNRRFJ
|
6.0 | Ki | 70 | — | |
DYSRECIVMDGUQU
|
6.0 | Ki | 29 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LYNBNVBMAGDJRW
|
6.0 | Ki | 81 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
VGWCJGBQHCMHNJ
|
6.0 | IC50 | 8 | — |