Target Details
| UniProt AC | Q9NR20 |
|---|---|
| Gene Symbol | DYRK4 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 139
- Clinical molecules 1
- Avg pChEMBL 6.45
Active Molecules (139)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJWUVVGOTOMGOH
|
6.5 | IC50 | 12 | — | |
UXUQVXDYXKMCGA
|
6.5 | Ki | 21 | — | |
JFDRONLMXPRQPP
|
6.5 | IC50 | 9 | — | |
OVVHFDIQCYTOAS
|
6.5 | IC50 | 9 | — | |
SJYQOVMGZOATNK
|
6.5 | IC50 | 9 | — | |
YORVMWUGDVGXOQ
|
6.5 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
6.5 | IC50 | 9 | — | |
IDOKKOQIQLHASZ
|
6.4 | IC50 | 8 | — | |
FIVWKNZKXNNFCW
|
6.4 | IC50 | 8 | — | |
OQSBQXVIMQMCES
|
6.4 | IC50 | 9 | — | |
BSFNGHCTZDCQBF
|
6.4 | Ki | 93 | — | |
CPGKMMMSMJKHDL
|
6.4 | Ki | 16 | — | |
MNVPCONHWCXDES
|
6.4 | IC50 | 9 | — | |
OWDRQHVEJIYVOI
|
6.4 | Ki | 47 | — | |
BWORFRWIDWQHPL
|
6.4 | IC50 | 7 | — | |
NBTJWRPKGNQBJS
|
6.4 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
6.4 | IC50 | 9 | — | |
QHTJZFWEQYRYQE
|
6.4 | IC50 | 9 | — | |
XTJRKTBELWGSDN
|
6.4 | IC50 | 8 | — | |
JBWDTSLHUJHODF
|
6.3 | IC50 | 9 | — | |
WQYUNADCLFWKGN
|
6.3 | IC50 | 7 | — | |
YDTHCIZMSQZYMR
|
6.3 | IC50 | 7 | — | |
BWKADHBOXYDZFU
|
6.3 | IC50 | 10 | — | |
SKKBUBMBPCJYKW
|
6.3 | IC50 | 9 | — | |
CLEGDJQQHUTCOW
|
6.3 | Ki | 43 | — | |
DCHAEDURAZJASA
|
6.3 | IC50 | 9 | — | |
UYJNQQDJUOUFQJ
|
6.3 | Ki | 68 | — | |
YMIJUBCSOKSFRU
|
6.3 | Ki | 87 | — | |
QTRZNDLLYHSJSH
|
6.3 | IC50 | 7 | — | |
YHZQZEGQCKWCLP
|
6.3 | IC50 | 9 | — | |
PGPHHJBZEGSUNE
|
6.3 | IC50 | 21 | — | |
PGPHHJBZEGSUNE
|
6.3 | IC50 | 17 | — | |
VCCCOYOXNKTQFO
|
6.3 | IC50 | 9 | — | |
FBURYRMHEHTVED
|
6.3 | IC50 | 9 | — | |
XTJRKTBELWGSDN
|
6.3 | IC50 | 8 | — | |
YDTHCIZMSQZYMR
|
6.3 | IC50 | 9 | — | |
DJHMDVUOYUYLOJ
|
6.2 | IC50 | 9 | — | |
JXQZHHAAJMQJKU
|
6.2 | IC50 | 9 | — | |
LXQXBEIFOYAXOP
|
6.2 | IC50 | 9 | — | |
ZFOMCSNUEHMROO
|
6.2 | IC50 | 7 | — | |
UGYUFJPHSWYELP
|
6.2 | IC50 | 8 | — | |
GXCOUFPTCZUTEE
|
6.2 | IC50 | 10 | — | |
RAQBQAXSLHDSKW
|
6.2 | IC50 | 8 | — | |
BPNUQXPIQBZCMR
|
6.2 | Ki | 60 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
LKUJDAHYLPICSE
|
6.2 | Ki | 24 | — | |
UMYSGMXAOXMMGG
|
6.2 | IC50 | 7 | — | |
YSBCFQVEEKUZSU
|
6.2 | IC50 | 9 | — | |
QCHDHJOEPUQALZ
|
6.2 | IC50 | 9 | — | |
YJKPCYDSZXIODK
|
6.2 | IC50 | 8 | — |