Target Details
| UniProt AC | Q9NR20 |
|---|---|
| Gene Symbol | DYRK4 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 139
- Clinical molecules 1
- Avg pChEMBL 6.45
Active Molecules (139)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BQWWOBKMDWACGC
|
8.7 | IC50 | 8 | — | |
RKUKAACYUCUJEE
|
8.0 | Ki | 58 | — | |
QAJPIJHWTGPUNZ
|
7.9 | Ki | 37 | — | |
KHVQTEBOVFILCQ
|
7.5 | IC50 | 10 | — | |
MIKAKZKNMYZLDX
|
7.4 | Ki | 42 | — | |
QIYXLIZWXGGKOO
|
7.3 | IC50 | 10 | — | |
DPDVVGCNUWGGRS
|
7.3 | IC50 | 10 | — | |
JJJSCYSPSKBQAX
|
7.3 | Ki | 34 | — | |
SLKHMZQUNIHINK
|
7.1 | IC50 | 10 | — | |
QTRZNDLLYHSJSH
|
7.1 | IC50 | 9 | — | |
BUDHVVXPBGMAPV
|
7.0 | IC50 | 11 | — | |
HEVBCYZPXGZFGS
|
6.9 | IC50 | 11 | — | |
IJFKKIMDRSZOOW
|
6.9 | IC50 | 9 | — | |
GEJSQZULGDKBQV
|
6.9 | IC50 | 8 | — | |
JCFJQIHDZHHMQT
|
6.9 | Ki | 42 | — | |
UMTWTCVTRDYHQQ
|
6.9 | Ki | 56 | — | |
YAXGFAAKCUOWNM
|
6.9 | IC50 | 9 | — | |
DXVSNYWBRDTHFF
|
6.9 | IC50 | 10 | — | |
SJWUVVGOTOMGOH
|
6.9 | IC50 | 10 | — | |
DCJOTKUJWJFCSP
|
6.8 | IC50 | 9 | — | |
QTRZNDLLYHSJSH
|
6.8 | IC50 | 9 | — | |
VCTLOEWZYIGVBO
|
6.8 | IC50 | 12 | — | |
YRFAWSIUIFNVQA
|
6.8 | IC50 | 9 | — | |
XPHWIERLJBFPFV
|
6.8 | Ki | 69 | — | |
NMUDZNRXZXDYEQ
|
6.8 | IC50 | 9 | — | |
CGPYAXSYKQBYKJ
|
6.8 | IC50 | 12 | — | |
SJWUVVGOTOMGOH
|
6.8 | IC50 | 9 | — | |
BULHRWBHKAVJMT
|
6.8 | IC50 | 8 | — | |
WREJZZXSNOJGIW
|
6.7 | IC50 | 9 | — | |
DKXHSOUZPMHNIZ
|
6.7 | Ki | 51 | Yes | |
SBYPANVVFZBWDF
|
6.7 | IC50 | 9 | — | |
YEZMGVBTPDYRPO
|
6.7 | IC50 | 8 | — | |
WFOMWAYINPJPDX
|
6.6 | IC50 | 9 | — | |
QXFBTYPBHYOEMX
|
6.6 | IC50 | 9 | — | |
YSODDCRKIDDXKM
|
6.6 | IC50 | 9 | — | |
PCQMERRARZKTPW
|
6.6 | Ki | 68 | — | |
YWTBGJGMTBHQTM
|
6.6 | Ki | 65 | — | |
MQRHLOPPMRFMKM
|
6.6 | IC50 | 9 | — | |
LVSVYVPFNYRNOF
|
6.6 | IC50 | 8 | — | |
QMUKOEKTUBVPFU
|
6.6 | IC50 | 12 | — | |
BWNQBFHVFFZHMR
|
6.6 | IC50 | 10 | — | |
FGBSSPMQGRUJPS
|
6.6 | IC50 | 10 | — | |
RJYLSCSDDDQEPD
|
6.5 | IC50 | 10 | — | |
MCNDTHVVURYHKT
|
6.5 | IC50 | 8 | — | |
OWDVXJJCVWTPPW
|
6.5 | IC50 | 8 | — | |
CHQYAWLKOUOTQO
|
6.5 | IC50 | 20 | — | |
AOGIFFVMTGMFBP
|
6.5 | IC50 | 8 | — | |
GCBJDOWIQHMCMR
|
6.5 | Ki | 84 | — | |
NJPWCTYVEJIQBM
|
6.5 | Ki | 72 | — | |
OWFLADWRSCINST
|
6.5 | Ki | 30 | — |