Target Details
| UniProt AC | Q9NQU5 |
|---|---|
| Gene Symbol | PAK6 |
| Protein Name | Serine/threonine-protein kinase PAK 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 21
- Clinical molecules 6
- Avg pChEMBL 7.23
KEGG Pathways (9)
Active Molecules (21)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.2 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
9.2 | Kd | 213 | — | |
PBCZSGKMGDDXIJ
|
8.4 | Kd | 68 | Yes | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
AYCPARAPKDAOEN
|
7.8 | IC50 | 73 | — | |
YFNWWNRZJGMDBR
|
7.7 | Kd | 35 | — | |
KGPGFQWBCSZGEL
|
7.7 | Kd | 59 | Yes | |
NXSJMRCTGYTSTK
|
7.7 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
RZXMIHOUHYSGJO
|
7.4 | IC50 | 4 | — | |
DGLFSNZWRYADFC
|
7.2 | IC50 | 12 | — | |
FPQNRXITKTZFMF
|
7.0 | Kd | 13 | — | |
ZCCPLJOKGAACRT
|
7.0 | Kd | 599 | — | |
LOLPPWBBNUVNQZ
|
6.7 | Kd | 97 | Yes | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
WINHZLLDWRZWRT
|
6.3 | Ki | 201 | Yes | |
BPNUQXPIQBZCMR
|
6.1 | Kd | 83 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |