Target Details
| UniProt AC | Q9NQS7 |
|---|---|
| Gene Symbol | INCENP |
| Protein Name | Inner centromere protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03941 (INCENP_ARK-bind) PF12178 (INCENP_N) |
Summary
- Multi-target molecules 93
- Clinical molecules 9
- Avg pChEMBL 7.1
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJQWORQRPDYKRS
|
6.8 | IC50 | 7 | — | |
HXAUJHZZPCBFPN
|
6.8 | IC50 | 4 | — | |
KTPMQAQBFZCIRN
|
6.8 | IC50 | 3 | — | |
YFBSBJBNKSZCLY
|
6.8 | IC50 | 4 | — | |
IABSWKZENVKESR
|
6.7 | IC50 | 3 | — | |
VTYQURZUYOUAOK
|
6.7 | IC50 | 3 | — | |
KUVJIFPAOJEBMN
|
6.7 | IC50 | 3 | — | |
LFVVQRUJKSZURN
|
6.7 | IC50 | 3 | — | |
WDVLOKNHMBINOL
|
6.7 | IC50 | 3 | — | |
ZWRIWNSRFLBBOD
|
6.7 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
6.7 | Kd | 1075 | — | |
WOMKQOXPOGODKV
|
6.7 | IC50 | 3 | — | |
GJDYHJPLCHRKEK
|
6.7 | IC50 | 3 | — | |
CHAZIKNZOXHZJA
|
6.6 | IC50 | 3 | — | |
CBBZXHUFHIEZHP
|
6.6 | IC50 | 4 | — | |
AOMMHIPSMLPJKQ
|
6.6 | IC50 | 4 | — | |
XTULNCWAJUYUIA
|
6.5 | IC50 | 4 | — | |
XZTYFGBEDWNFPM
|
6.5 | IC50 | 3 | — | |
RPMDNLSTGYONBC
|
6.5 | IC50 | 3 | — | |
PMDUMOUXISSZED
|
6.4 | IC50 | 3 | — | |
DQPVIVGCZVQZDO
|
6.4 | IC50 | 3 | — | |
LKZXAQZZOSZHLE
|
6.4 | IC50 | 3 | — | |
AFPQNJFINOFINI
|
6.3 | IC50 | 3 | — | |
LLROFEFDEFKWQN
|
6.3 | IC50 | 3 | — | |
UVHDAKLRGJSVKQ
|
6.2 | IC50 | 4 | — | |
DUKJABPGWUISRC
|
6.2 | IC50 | 3 | — | |
ULDURKNHYFYKMS
|
6.2 | IC50 | 3 | — | |
GPPDWFNQVHJOEU
|
6.2 | IC50 | 3 | — | |
IDKYOQDTCCUVIN
|
6.2 | IC50 | 3 | — | |
USUYXDKUCNQBKM
|
6.2 | IC50 | 3 | — | |
MNYJXBQMADDOQS
|
6.2 | IC50 | 3 | — | |
TWPZRFZCHZSVKG
|
6.1 | IC50 | 4 | — | |
GABKCBKPNYHAJC
|
6.1 | IC50 | 3 | — | |
WROHCHCGJIWAPG
|
6.1 | IC50 | 3 | — | |
FATFDRYYCYZBQB
|
6.1 | IC50 | 5 | Yes | |
IMQVBCRZLIQNPG
|
6.1 | IC50 | 5 | Yes | |
LZKFDPIUYGTKHZ
|
6.1 | IC50 | 3 | — | |
WFJYZRKNRWYRTN
|
6.1 | IC50 | 3 | — | |
WWPZBBQLQAEXGE
|
6.1 | IC50 | 3 | — | |
UVHDAKLRGJSVKQ
|
6.1 | IC50 | 3 | — | |
ZGCQIBQYASDQPM
|
6.1 | IC50 | 3 | — | |
AFPQNJFINOFINI
|
6.0 | IC50 | 4 | — | |
GBAHUNGQGRGJAX
|
6.0 | IC50 | 3 | — |