Target Details
| UniProt AC | Q9NQS7 |
|---|---|
| Gene Symbol | INCENP |
| Protein Name | Inner centromere protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03941 (INCENP_ARK-bind) PF12178 (INCENP_N) |
Summary
- Multi-target molecules 93
- Clinical molecules 9
- Avg pChEMBL 7.1
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULOLUGXMKLIZGE
|
9.3 | IC50 | 8 | Yes | |
WKDACQVEJIVHMZ
|
9.3 | IC50 | 46 | — | |
QWJHWNIFEWOQTF
|
9.2 | IC50 | 5 | Yes | |
ZLHFILGSQDJULK
|
9.0 | IC50 | 37 | Yes | |
QTBWCSQGBMPECM
|
8.8 | Ki | 21 | Yes | |
CZVVMRNEBRFYTL
|
8.7 | IC50 | 9 | Yes | |
QNOOVTZVMOOSAW
|
8.5 | IC50 | 4 | — | |
BRXHKUKMMZTVRE
|
8.4 | IC50 | 3 | — | |
RBMOLIOJAWRTIV
|
8.4 | IC50 | 4 | — | |
ZLODPJRHCQWJSX
|
8.4 | IC50 | 3 | — | |
CDQHQPMNSRRDJP
|
8.2 | IC50 | 3 | — | |
DSLKQMBMFBKGRK
|
8.2 | IC50 | 4 | — | |
MENIKIFJGYYVNI
|
8.2 | IC50 | 5 | Yes | |
MTPMSKFDRZNUFI
|
8.2 | IC50 | 3 | — | |
WVYZESHCWKLDBS
|
8.2 | IC50 | 5 | Yes | |
NNZRYGISYKGSCW
|
8.1 | IC50 | 3 | — | |
RBMOLIOJAWRTIV
|
8.1 | IC50 | 5 | — | |
VPEYPVPNDMIFEL
|
8.0 | IC50 | 3 | — | |
KBNSMUBNIUALHR
|
7.9 | IC50 | 3 | — | |
JWILUIVAYLRFIY
|
7.7 | IC50 | 14 | — | |
DUAVMQAFJJEDTP
|
7.7 | IC50 | 3 | — | |
LCVIRAZGMYMNNT
|
7.6 | IC50 | 20 | — | |
HQTDBFXCCUUCFU
|
7.6 | IC50 | 2 | — | |
ZDDITUPJXGNNKU
|
7.5 | IC50 | 3 | — | |
ASVHLUISRWYGFL
|
7.5 | IC50 | 3 | — | |
RHELVXGNWNTPJF
|
7.4 | IC50 | 3 | — | |
XEADJJXUBNVGAN
|
7.4 | IC50 | 3 | — | |
VHSSUFWQNFHOQT
|
7.4 | IC50 | 3 | — | |
WBOJNPOFWWQXBX
|
7.4 | IC50 | 4 | — | |
DXXQAWREKCQJCS
|
7.3 | IC50 | 4 | — | |
ROPCWFYJUONUHM
|
7.3 | IC50 | 4 | — | |
SIRZTYWYVGTPEV
|
7.3 | IC50 | 4 | — | |
FLGUGRAWIWHCJF
|
7.3 | IC50 | 4 | — | |
OSVOVHIYXDNBJQ
|
7.3 | IC50 | 3 | — | |
FJZFOTKMZCYJDF
|
7.2 | IC50 | 4 | — | |
IRGIWNWHHPMOLO
|
7.2 | IC50 | 3 | — | |
PZWGYFJPWNXLGT
|
7.2 | IC50 | 3 | — | |
BMYPVSWCQCKWHI
|
7.2 | IC50 | 3 | — | |
CQOOBCLBMYGVDE
|
7.2 | IC50 | 3 | — | |
KLIDFKYRDXZCOP
|
7.1 | IC50 | 4 | — | |
IYBGHBZUXSMOKI
|
7.0 | IC50 | 3 | — | |
GXKIHPXGVQZMIN
|
7.0 | IC50 | 3 | — | |
ROJRDYDJKQGLRH
|
7.0 | IC50 | 3 | — | |
DADASRPKWOGKCU
|
7.0 | IC50 | 9 | — | |
ODIUNKSOMOLOOF
|
7.0 | IC50 | 3 | — | |
YGEQQFLMLXRDQK
|
6.9 | IC50 | 3 | — | |
ARLBCCDWOPSKDJ
|
6.9 | IC50 | 3 | — | |
MCVWAVHQVAZAKZ
|
6.9 | IC50 | 3 | — | |
WOSUZOOSGPAWAC
|
6.9 | IC50 | 3 | — | |
YAEXRFPBDXLXMG
|
6.8 | IC50 | 3 | — |