Target Details
| UniProt AC | Q9NQB0 |
|---|---|
| Gene Symbol | TCF7L2 |
| Protein Name | Transcription factor 7-like 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08347 (CTNNB1_binding) PF00505 (HMG_box) |
Summary
- Multi-target molecules 154
- Clinical molecules 0
- Avg pChEMBL 6.29
KEGG Pathways (21)
- Acute myeloid leukemia
- Adherens junction
- Alcoholic liver disease
- Arrhythmogenic right ventricular cardiomyopathy
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Colorectal cancer
- Cushing syndrome
- Endometrial cancer
- Gastric cancer
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human papillomavirus infection
- Kaposi sarcoma-associated herpesvirus infection
- Melanogenesis
- Pathways in cancer
- Prostate cancer
- Salmonella infection
- Thyroid cancer
- Wnt signaling pathway
Associated Diseases (1)
Active Molecules (154)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JIFZTSSDQGCLLR
|
6.1 | IC50 | 2 | — | |
JKXMHWLJTNPRNY
|
6.1 | IC50 | 2 | — | |
OWBJDMRAJLJHRC
|
6.1 | IC50 | 2 | — | |
GALPVVQJEKJSTD
|
6.1 | IC50 | 2 | — | |
LNJYCOSDXHETRQ
|
6.1 | IC50 | 2 | — | |
WVCVWOPBLAPLQC
|
6.1 | IC50 | 2 | — | |
BJCUXRXFKGWVII
|
6.1 | IC50 | 2 | — | |
CCWKJFUTAIMLPZ
|
6.1 | IC50 | 2 | — | |
LCIVGEQOKDTWOD
|
6.1 | IC50 | 2 | — | |
UQOAIOXRQHVEGJ
|
6.1 | IC50 | 2 | — | |
KAMBUPZZPWFSKM
|
6.1 | IC50 | 2 | — | |
GOZXIWWTPDNZDG
|
6.1 | IC50 | 2 | — | |
HENJNCNHECLTNG
|
6.1 | IC50 | 2 | — | |
PZPRCQDQUVGRPJ
|
6.1 | IC50 | 2 | — | |
YOTKDEFXCGRSLS
|
6.1 | IC50 | 2 | — | |
BTXSPVOFVGXDFM
|
6.1 | IC50 | 2 | — | |
LDHXAKDEJVSJPT
|
6.1 | IC50 | 2 | — | |
OIKBHWKMMTUEMF
|
6.1 | IC50 | 2 | — | |
WTYQIOUFJVYAIT
|
6.1 | IC50 | 2 | — | |
BUTHRHISDJBKQI
|
6.1 | IC50 | 2 | — | |
JXOBVBGRETYJJP
|
6.1 | IC50 | 2 | — | |
PFXNWGOEZFFOCP
|
6.1 | IC50 | 2 | — | |
PZGNGHTYQPXUTG
|
6.1 | IC50 | 2 | — | |
SEEGTULJFJHBLM
|
6.1 | IC50 | 2 | — | |
UEDRGVUEMGGOSD
|
6.1 | IC50 | 2 | — | |
AAWMPINFKWIDEX
|
6.1 | IC50 | 2 | — | |
HKSDCISEGHSAGG
|
6.1 | IC50 | 2 | — | |
HWPXDAIDFOHAOQ
|
6.1 | IC50 | 2 | — | |
GGGBVFZOZOBFCR
|
6.1 | IC50 | 2 | — | |
HIKINKJOKJCOLS
|
6.1 | IC50 | 2 | — | |
LGSPOEDRBUBJBK
|
6.1 | IC50 | 2 | — | |
SOZJMQJCCKPSJW
|
6.1 | IC50 | 2 | — | |
UINJQSGTMGWCGS
|
6.1 | IC50 | 2 | — | |
XHLPHDKEOZRIGH
|
6.1 | IC50 | 2 | — | |
DCANTODNDYGXLJ
|
6.0 | IC50 | 2 | — | |
NJKQOFYYUWSENG
|
6.0 | IC50 | 2 | — | |
VALDLJHSDBHIOB
|
6.0 | IC50 | 2 | — | |
DLOBJTOTFRGFMG
|
6.0 | IC50 | 2 | — | |
DTQNBUHVSZINJH
|
6.0 | IC50 | 2 | — | |
RRZIAHBPWFIHEA
|
6.0 | IC50 | 2 | — | |
YMODINPCEMVPDZ
|
6.0 | IC50 | 2 | — | |
CICSICZXJDAQLA
|
6.0 | IC50 | 2 | — | |
FDQIPUBUNUJHCQ
|
6.0 | IC50 | 2 | — | |
RQMISRRRFAECOZ
|
6.0 | IC50 | 2 | — | |
SPDURWZIHZPWCS
|
6.0 | IC50 | 2 | — | |
CODWCDWXNSITLV
|
6.0 | IC50 | 2 | — | |
FKUFZNJYPFAVRD
|
6.0 | IC50 | 2 | — | |
JGVVMIZDHYWMPF
|
6.0 | IC50 | 2 | — | |
ALUJTNZFYZSCHV
|
6.0 | IC50 | 2 | — | |
DCXKFVRAFWMNLE
|
6.0 | IC50 | 2 | — |