Target Details
| UniProt AC | Q9NQB0 |
|---|---|
| Gene Symbol | TCF7L2 |
| Protein Name | Transcription factor 7-like 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08347 (CTNNB1_binding) PF00505 (HMG_box) |
Summary
- Multi-target molecules 154
- Clinical molecules 0
- Avg pChEMBL 6.29
KEGG Pathways (21)
- Acute myeloid leukemia
- Adherens junction
- Alcoholic liver disease
- Arrhythmogenic right ventricular cardiomyopathy
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Colorectal cancer
- Cushing syndrome
- Endometrial cancer
- Gastric cancer
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human papillomavirus infection
- Kaposi sarcoma-associated herpesvirus infection
- Melanogenesis
- Pathways in cancer
- Prostate cancer
- Salmonella infection
- Thyroid cancer
- Wnt signaling pathway
Associated Diseases (1)
Active Molecules (154)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WWBNWNFPDKAYDJ
|
6.4 | IC50 | 2 | — | |
ZCFCGIVOFXMJEF
|
6.4 | IC50 | 2 | — | |
RNIJMIWIFOAASJ
|
6.4 | IC50 | 2 | — | |
YAPPCPXCPKDGIM
|
6.4 | IC50 | 2 | — | |
DXTSVDRTSAEVPU
|
6.3 | IC50 | 2 | — | |
JJEDWBQZCRESJL
|
6.3 | Kd | 3 | — | |
MWXNTFWHXGUHAA
|
6.3 | IC50 | 2 | — | |
XDTNFQZQMHHVRT
|
6.3 | IC50 | 2 | — | |
BCUICGCNNXVMLE
|
6.3 | IC50 | 2 | — | |
OTSATXCTGPMHFD
|
6.3 | IC50 | 2 | — | |
REZMBQZQTXXSMK
|
6.3 | IC50 | 2 | — | |
JYCJFPNHRMLHDX
|
6.3 | IC50 | 2 | — | |
CKWRKEGEENQUQW
|
6.3 | IC50 | 2 | — | |
PBBVEJYBMVJMJF
|
6.3 | IC50 | 2 | — | |
MZGDZKMEBPEZSZ
|
6.3 | IC50 | 2 | — | |
QBRMWVWITQHRJX
|
6.3 | IC50 | 2 | — | |
BAHPJNWHTFCKKZ
|
6.3 | IC50 | 2 | — | |
GSADWJIOPNLJGU
|
6.3 | IC50 | 2 | — | |
QYLLEMWBHJWWNX
|
6.3 | IC50 | 2 | — | |
SWHPJPYLDRQPFW
|
6.3 | IC50 | 2 | — | |
ZBNFPOPNAPVGTL
|
6.3 | IC50 | 2 | — | |
GXJWTRQQFNHPOC
|
6.3 | IC50 | 2 | — | |
RGFXAEWWEUXTCN
|
6.3 | IC50 | 2 | — | |
YMPDOPQOELVBID
|
6.3 | IC50 | 2 | — | |
LBWYBHYHBIMHKK
|
6.3 | IC50 | 2 | — | |
KNYUKCDFZOGMCJ
|
6.3 | IC50 | 2 | — | |
QYLLEMWBHJWWNX
|
6.3 | IC50 | 2 | — | |
HRAUHIORVNXMMW
|
6.2 | IC50 | 2 | — | |
LBWYBHYHBIMHKK
|
6.2 | IC50 | 2 | — | |
MHBWTTBCDCFUFG
|
6.2 | IC50 | 2 | — | |
JHFRHTLCCWDGCE
|
6.2 | IC50 | 2 | — | |
BHIOLGCZMCCQKQ
|
6.2 | IC50 | 2 | — | |
FIIDIYQVDYCCRC
|
6.2 | IC50 | 2 | — | |
FTPFZJMAJIPMNS
|
6.2 | IC50 | 2 | — | |
GSIFXTHXPURSBY
|
6.2 | IC50 | 2 | — | |
IVGZYIDZKCELCR
|
6.2 | IC50 | 2 | — | |
NBQAGLPJFGLCAC
|
6.2 | IC50 | 2 | — | |
RGPXAJSDCKQSRK
|
6.2 | IC50 | 2 | — | |
WKVYSKUPYSAOHQ
|
6.2 | IC50 | 2 | — | |
PIROHBFQHMKAPE
|
6.2 | IC50 | 2 | — | |
CSQCUQGTDYPDOZ
|
6.2 | IC50 | 2 | — | |
YUFYCCNECIZYEE
|
6.2 | IC50 | 2 | — | |
ZAKBAQHYORKWNL
|
6.2 | IC50 | 2 | — | |
ARYMNZXRDFPPLP
|
6.2 | IC50 | 2 | — | |
LLKZNBPLCIOFFO
|
6.2 | IC50 | 2 | — | |
OXVKTAYGDZEXJL
|
6.2 | IC50 | 2 | — | |
WNJZFQIJHPAMLL
|
6.2 | IC50 | 2 | — | |
MDSQKPYZQOGJBG
|
6.2 | IC50 | 2 | — | |
XCVHXLUZZXQNPB
|
6.2 | IC50 | 2 | — | |
FDBTXMURTPTNCO
|
6.1 | IC50 | 2 | — |