Target Details
| UniProt AC | Q9NQB0 |
|---|---|
| Gene Symbol | TCF7L2 |
| Protein Name | Transcription factor 7-like 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08347 (CTNNB1_binding) PF00505 (HMG_box) |
Summary
- Multi-target molecules 154
- Clinical molecules 0
- Avg pChEMBL 6.29
KEGG Pathways (21)
- Acute myeloid leukemia
- Adherens junction
- Alcoholic liver disease
- Arrhythmogenic right ventricular cardiomyopathy
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Colorectal cancer
- Cushing syndrome
- Endometrial cancer
- Gastric cancer
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human papillomavirus infection
- Kaposi sarcoma-associated herpesvirus infection
- Melanogenesis
- Pathways in cancer
- Prostate cancer
- Salmonella infection
- Thyroid cancer
- Wnt signaling pathway
Associated Diseases (1)
Active Molecules (154)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
COJZCIROPCHMHD
|
7.0 | IC50 | 2 | — | |
QMMLHHLWVXDIKW
|
6.9 | IC50 | 2 | — | |
UFDQFCNUXSHUFA
|
6.9 | IC50 | 2 | — | |
ZSNPUIWMTSJNFC
|
6.8 | IC50 | 2 | — | |
AHCNMJSYWNOADJ
|
6.8 | IC50 | 2 | — | |
MAISCMHHSMCHBZ
|
6.7 | IC50 | 2 | — | |
OWFZSPWWASOCHH
|
6.7 | IC50 | 2 | — | |
GOGYIQLIDQSVSG
|
6.7 | IC50 | 2 | — | |
JMWWPTLJPVTWTM
|
6.7 | IC50 | 2 | — | |
SACAWJSUCOAUFA
|
6.7 | IC50 | 2 | — | |
VIEVQOCWEOSVBZ
|
6.7 | IC50 | 2 | — | |
NMWAOZPEEIODED
|
6.7 | IC50 | 2 | — | |
AOCHSTRFBNLJOW
|
6.6 | IC50 | 2 | — | |
KPQJQZXAXPLRFI
|
6.6 | IC50 | 2 | — | |
OLKDOXDHHWVAQT
|
6.6 | IC50 | 2 | — | |
MWXNTFWHXGUHAA
|
6.6 | IC50 | 2 | — | |
DLPHGOYOYJSYIG
|
6.6 | IC50 | 2 | — | |
XUHLUGUZGFIDEE
|
6.5 | IC50 | 2 | — | |
AQNZWUSOYZCMEB
|
6.5 | IC50 | 2 | — | |
SNAKNDOGCPAEQI
|
6.5 | IC50 | 2 | — | |
UCEGDYDPOSBUTP
|
6.5 | IC50 | 6 | — | |
MNDIKUFVYLXDTF
|
6.5 | IC50 | 2 | — | |
WIKFZOQKGJIUSK
|
6.5 | IC50 | 2 | — | |
YEWKMXVZMMJARV
|
6.5 | IC50 | 2 | — | |
FPGLHUFTBYVZPN
|
6.5 | IC50 | 2 | — | |
IJLBBQLZALRRRA
|
6.5 | IC50 | 2 | — | |
WVEQLRDSEPTHHS
|
6.5 | IC50 | 2 | — | |
CTLKHRIZXUQDGT
|
6.5 | IC50 | 2 | — | |
QNSYZPLZZGYLQU
|
6.5 | IC50 | 2 | — | |
QWNBSJOCJVHVKS
|
6.5 | IC50 | 2 | — | |
BKVYPGMSWDCQQJ
|
6.5 | IC50 | 2 | — | |
DZXTZSYPFBOUDK
|
6.5 | IC50 | 2 | — | |
KEPNWCPTSUWOJV
|
6.5 | IC50 | 2 | — | |
SNCNFKSRYUUHAW
|
6.5 | IC50 | 2 | — | |
WLIFRFDORDZAFM
|
6.4 | IC50 | 2 | — | |
FDVIIYLZXNBDQS
|
6.4 | IC50 | 2 | — | |
CSEZGDFMVUEWID
|
6.4 | IC50 | 2 | — | |
CSQCUQGTDYPDOZ
|
6.4 | IC50 | 2 | — | |
FUIUGMVSXLFMNI
|
6.4 | IC50 | 2 | — | |
HBXAFXUIBLVCRO
|
6.4 | IC50 | 2 | — | |
LKDLIWZRZLKJNX
|
6.4 | IC50 | 2 | — | |
NGLYERQRYRDLCH
|
6.4 | IC50 | 2 | — | |
LRLFSSDGEWJOLP
|
6.4 | IC50 | 2 | — | |
ZAARNDKEWLKRPI
|
6.4 | IC50 | 2 | — | |
FDVIIYLZXNBDQS
|
6.4 | IC50 | 2 | — | |
WLBYUHHEOYDONA
|
6.4 | IC50 | 2 | — | |
MHNXYZVWDASRHS
|
6.4 | IC50 | 2 | — | |
CXCCXQJROQTCHJ
|
6.4 | IC50 | 2 | — | |
LDNKLYQETCREAU
|
6.4 | IC50 | 2 | — | |
NKYVJKPVWKBETD
|
6.4 | IC50 | 2 | — |