Target Details
| UniProt AC | Q9NPI1 |
|---|---|
| Gene Symbol | BRD7 |
| Protein Name | Bromodomain-containing protein 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF12024 (DUF3512) |
Summary
- Multi-target molecules 28
- Clinical molecules 0
- Avg pChEMBL 6.74
KEGG Pathways (2)
Active Molecules (28)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UOQAFGWMKNIVAR
|
9.1 | Kd | 6 | — | |
HONYBLSJNSYWKQ
|
7.6 | Ki | 3 | — | |
JSTVWXBDEJQXEC
|
7.4 | IC50 | 2 | — | |
BMVCSXFOQPYKKC
|
7.1 | IC50 | 5 | — | |
PMWIFIWWNULSSP
|
7.0 | Kd | 2 | — | |
UIULTDHSORWSLL
|
7.0 | IC50 | 2 | — | |
FWTDDBIMDSVPTR
|
7.0 | Kd | 2 | — | |
RBUYFHLQNPJMQM
|
6.9 | Kd | 10 | — | |
AWVPNUWHMBPXOU
|
6.9 | Kd | 8 | — | |
BJFSUDWKXGMUKA
|
6.9 | Kd | 3 | — | |
UEMQPCYDWCSVCU
|
6.8 | IC50 | 5 | — | |
SZKYAPUMPFTJEP
|
6.7 | IC50 | 2 | — | |
JGOZUFGBTSAWEI
|
6.7 | Kd | 4 | — | |
DBVNJIZWSYAIOO
|
6.6 | Kd | 7 | — | |
OAXPZAPALNMAIG
|
6.6 | IC50 | 2 | — | |
GQTWFQWDINXZPP
|
6.6 | IC50 | 2 | — | |
WCRAZRPWWUJMQW
|
6.5 | Ki | 2 | — | |
GVJYOLRRZZUUOE
|
6.5 | Kd | 5 | — | |
RPBMXJHQYJLPDN
|
6.5 | Kd | 2 | — | |
LBUBPCSKFDKKFO
|
6.4 | Kd | 2 | — | |
UYBRROMMFMPJAN
|
6.4 | Kd | 8 | — | |
WRUWGLUCNBMGPS
|
6.4 | Kd | 5 | — | |
DGJREYHVQYZTEV
|
6.4 | Kd | 6 | — | |
UXFKGTAATGRBOW
|
6.3 | Ki | 2 | — | |
QVMOJFHRHLLSOT
|
6.3 | Kd | 3 | — | |
QCIJLRJBZDBVDB
|
6.1 | Kd | 5 | — | |
ZJBYPBSYPDAGHO
|
6.1 | Ki | 2 | — | |
LVDRREOUMKACNJ
|
6.0 | Kd | 2 | — |