Target Details
| UniProt AC | Q9HCP0 |
|---|---|
| Gene Symbol | CSNK1G1 |
| Protein Name | Casein kinase I isoform gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12605 (CK1gamma_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 99
- Clinical molecules 7
- Avg pChEMBL 6.65
KEGG Pathways (1)
Active Molecules (99)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMIJUBCSOKSFRU
|
6.5 | Ki | 87 | — | |
BPNUQXPIQBZCMR
|
6.4 | Ki | 60 | — | |
HEKAIDKUDLCBRU
|
6.4 | Ki | 20 | — | |
IQNOGQGSOHNMCL
|
6.4 | Ki | 14 | — | |
SPOBBSBKXJKGBG
|
6.4 | Ki | 16 | — | |
GQHMZZXJWGPHDA
|
6.3 | Ki | 20 | — | |
KXPWWMPXNUOYOH
|
6.3 | Ki | 24 | — | |
MTYMWGNJKDHWGN
|
6.3 | Ki | 18 | — | |
BPNUQXPIQBZCMR
|
6.3 | Kd | 83 | Yes | |
SOUYYRXENUITFU
|
6.3 | IC50 | 2 | — | |
KQWTXAWKBUUOMU
|
6.2 | IC50 | 20 | Yes | |
BIKYDWLMTPRSQL
|
6.2 | Ki | 50 | — | |
CLRFYTGANQZOBS
|
6.2 | Ki | 41 | — | |
DPPIQOOVRLCHQC
|
6.2 | Ki | 6 | — | |
KAKFXRYHYUPXSU
|
6.2 | Ki | 16 | — | |
MIKAKZKNMYZLDX
|
6.2 | Ki | 42 | — | |
MVJMMLFMPWITEJ
|
6.2 | Ki | 110 | — | |
ULHGAQSVFPOUDY
|
6.2 | Ki | 43 | — | |
UVZVWLFSZNPMBS
|
6.2 | Ki | 17 | — | |
XJJYJNMNYDNXNO
|
6.2 | Ki | 23 | — | |
DKZYXHCYPUVGAF
|
6.2 | Kd | 112 | — | |
AOFJRBMLTUGMMP
|
6.1 | Ki | 12 | — | |
GEGCXGMFUYJULA
|
6.1 | Ki | 30 | Yes | |
GUMBHNMWKMFKRT
|
6.1 | Ki | 23 | — | |
GWMATETWMAQOFL
|
6.1 | Ki | 36 | — | |
MGNQNQOSSLCUFP
|
6.1 | Ki | 12 | — | |
UTMRCMCLMBDPNW
|
6.1 | Ki | 10 | — | |
VBIYDORVDCFKHM
|
6.1 | Ki | 13 | — | |
XBAIEEJJCJHBDL
|
6.1 | Ki | 17 | — | |
XYZNKCSDQRKAFR
|
6.1 | Ki | 53 | — | |
ZPVLRSVLOWVDJC
|
6.1 | Ki | 14 | — | |
HFNKQEVNSGCOJV
|
6.1 | Kd | 65 | — | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
CTNPALGJUAXMMC
|
6.0 | Kd | 151 | — | |
DZSUJUOJJJCWGG
|
6.0 | Ki | 55 | Yes | |
HOBMVEVXDIOMDM
|
6.0 | Ki | 18 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JZTOUVBEZONDKA
|
6.0 | Ki | 80 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KYACBMRLQMEIAI
|
6.0 | Ki | 30 | — | |
LGHBDVLAHHANMX
|
6.0 | Ki | 53 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
ODPGGGTTYSGTGO
|
6.0 | Kd | 153 | — | |
PQNWNVWJXPSZFR
|
6.0 | Ki | 21 | — | |
PYQFQGXOARMGAQ
|
6.0 | IC50 | 11 | — | |
TZSJMSZEKQGCBI
|
6.0 | Ki | 15 | — | |
WINHZLLDWRZWRT
|
6.0 | Ki | 66 | — | |
XSDJOIOVIMPMHD
|
6.0 | Ki | 44 | — | |
YEPNVBNYCRGZRX
|
6.0 | Ki | 26 | — |