Target Details
UniProt ACQ9HCP0
Gene SymbolCSNK1G1
Protein NameCasein kinase I isoform gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF12605 (CK1gamma_C) PF00069 (Pkinase)
Summary
  • Multi-target molecules 99
  • Clinical molecules 7
  • Avg pChEMBL 6.65
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (99)
InChIKey pChEMBL Type Targets Clinical
MUOKSQABCJCOPU 8.4 IC50 36
NWAUBAGBGOPJLF 8.4 Ki 51 Yes
SBFPHSVZEXSHTL 7.9 Ki 62
UDFDIIVNIYWXDM 7.8 Ki 74
XFWUTMHVDGPWLH 7.8 Ki 75
GNZPMJDEUIVORU 7.7 Ki 3
IMMZLRQJNZSTTE 7.7 Ki 15
ISVHLTLEHRZKJC 7.7 Ki 19
MFMXAWQGPQXDRJ 7.7 Ki 27
OBHNPUMYQHGYJJ 7.7 Ki 4
ROPVGAMDOWWUTK 7.7 Ki 5
RYAVJHIPOWNWDE 7.7 Ki 38
YKJSWMAVAKRUAN 7.7 Ki 19
RKUKAACYUCUJEE 7.6 Ki 58
ZGZVRPRSFXRGCF 7.6 Ki 76
KOHNRDPXFDZZJF 7.5 Ki 31
ATBAETXFFCOZOY 7.5 IC50 39
VGURQCQNQDZAOF 7.4 Ki 6
YWTBGJGMTBHQTM 7.4 Ki 65
QAJPIJHWTGPUNZ 7.3 Ki 37
CFDCGXXHXUZSNP 7.2 Kd 4
LXVBELDBJGYFEM 7.2 Ki 20
UMTWTCVTRDYHQQ 7.2 Ki 56
JJJSCYSPSKBQAX 7.1 Ki 34
NJPWCTYVEJIQBM 7.1 Ki 72
UTFXYGYVDDLJER 7.1 Ki 36
ADMFLILDQJSEIK 7.0 Ki 72
GCBJDOWIQHMCMR 7.0 Ki 84
CHTMRWQLNNRRFJ 6.9 Ki 70
CLEGDJQQHUTCOW 6.9 Ki 43
ASNQMAVHHGGQRB 6.8 Ki 14
GPXKVULNYYNGDP 6.8 IC50 4
LYNBNVBMAGDJRW 6.8 Ki 81
NEWAULHLLUCDPD 6.8 Ki 27
SYLTYCLPHHSEIJ 6.8 Ki 27
ZCCPLJOKGAACRT 6.6 Kd 599
DKXHSOUZPMHNIZ 6.6 Ki 51 Yes
IMHKMKWSWHFKTM 6.6 Ki 13
MCBPNFWHHNJTGN 6.6 IC50 5
OWFLADWRSCINST 6.6 Ki 30
VXYDJXMHISGSDA 6.6 Ki 59
XCHWBXBDZRJVDP 6.6 Ki 51
XDJCLCLBSGGNKS 6.5 Kd 21
DPDZHVCKYBCJHW 6.5 IC50 11
FUMCKNCUEAQHCV 6.5 Ki 103
HWGZXYUOXGVACR 6.5 Ki 6
ISEDKXOMRIKZPK 6.5 Ki 13
LCKDESRGCHSHHO 6.5 Ki 18
NLUPJKQOKWBWFC 6.5 Ki 69
XPHWIERLJBFPFV 6.5 Ki 69
2D structure