Target Details
UniProt ACQ9HBW0
Gene SymbolLPAR2
Protein NameLysophosphatidic acid receptor 2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 33
  • Clinical molecules 0
  • Avg pChEMBL 7.05
Top Co-occurrence Targets
Active Molecules (33)
InChIKey pChEMBL Type Targets Clinical
VEAJEWXYGKUGPH 8.2 IC50 4
HZFPOTBCYPWQSH 8.1 IC50 2
YIZUZSSLYPDFOC 7.8 IC50 4
WTJGTMFQALCKRT 7.7 IC50 4
SKDIMRRKRVTENP 7.7 IC50 2
GCTZIVJBMHYJOP 7.6 IC50 4
HXDPHSXYLHIVSE 7.6 IC50 4
DQXSYKMXKITFAL 7.5 IC50 3
SQBXAXYMXPCNON 7.4 IC50 4
IYOGKTIRIRHPOH 7.4 IC50 6
FSCOADFARBASQU 7.4 IC50 4
UVRGHEYADYBWFL 7.4 IC50 2
PCBMXZQDEQINJG 7.3 IC50 4
GBAYNJCGVHFQTM 7.2 IC50 4
YFWUAIPFVJAYCH 7.2 IC50 4
MMKMRZFTPGRQEQ 7.1 IC50 4
WECRLAZSZWCWDE 7.1 IC50 5
LYZKFLGVDKUPAP 7.0 IC50 4
BPRNMVDTWIHULJ 7.0 IC50 6
SHISURVONRMBAW 6.9 IC50 4
VKXANKHCILEVSX 6.9 IC50 4
HLVKVWDSLLFMSX 6.8 Ki 4
JGCATLCTRCCGRP 6.8 Ki 4
NSEVTFLGGHULPD 6.6 IC50 4
WFMGEMPWKRJJHM 6.6 IC50 3
JNAQEIPNFVZKSC 6.6 IC50 4
AEFXZQBYWHGBOY 6.5 IC50 2
KSAATBXYGYJAQU 6.4 IC50 4
AXAGGQQXMQHIFF 6.3 IC50 4
BDZJQGMIIWGSHK 6.3 IC50 4
POPQMXAKAVJFNJ 6.2 IC50 4
RDMIFINBVKZJSN 6.1 Ki 2
DAOODVJVNUBOQM 6.1 IC50 2
2D structure