Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAVINHSQSZLJGI
|
6.9 | IC50 | 2 | — | |
WPXVVAWAHQHJPF
|
6.9 | IC50 | 41 | — | |
BDNVJOGXLGPBFH
|
6.9 | IC50 | 2 | — | |
LJQCFLSZUSTALC
|
6.9 | IC50 | 2 | — | |
UWKJXDSZQTXARH
|
6.9 | IC50 | 2 | — | |
ZROBKNPXIOQRBD
|
6.8 | IC50 | 2 | — | |
HIPFDFQYWKJHND
|
6.8 | IC50 | 2 | — | |
CMWRPDHVGMHLSZ
|
6.8 | IC50 | 22 | — | |
QMEZKJBCLUGJTN
|
6.8 | IC50 | 5 | — | |
QMEZKJBCLUGJTN
|
6.8 | IC50 | 4 | — | |
AOBLBPWPSKBHSI
|
6.8 | Ki | 55 | — | |
CZIGMBNEFWBEMD
|
6.8 | Ki | 16 | — | |
DWXUTKBSWVUPBE
|
6.8 | Ki | 8 | — | |
GFYFRPOVKHGTOX
|
6.8 | IC50 | 2 | — | |
IZAVTOABECKIDH
|
6.8 | Ki | 20 | — | |
KJZWOUQMPQCYIK
|
6.8 | IC50 | 2 | — | |
LRLDYTTWQIFWBD
|
6.8 | Ki | 25 | — | |
NWAUBAGBGOPJLF
|
6.8 | Ki | 51 | Yes | |
SGVAIMLQDSZAQH
|
6.8 | IC50 | 2 | — | |
UFMAIBLTWQRHAK
|
6.8 | Ki | 10 | — | |
XFWUTMHVDGPWLH
|
6.8 | Ki | 75 | — | |
XOOAAYRIVATZNM
|
6.8 | Ki | 55 | — | |
NXSJMRCTGYTSTK
|
6.8 | Kd | 200 | — | |
OGDZDXFTNNLXFS
|
6.8 | IC50 | 2 | — | |
RYUUMGNHANZHLX
|
6.8 | Ki | 2 | — | |
TXTJPVXASVJOMW
|
6.8 | IC50 | 2 | — | |
DKXHSOUZPMHNIZ
|
6.8 | IC50 | 51 | Yes | |
LPDCQOLOXLFVBW
|
6.8 | IC50 | 2 | — | |
WHDVHWQDQBHJEN
|
6.8 | IC50 | 2 | — | |
WZILQEFHQBNHBB
|
6.8 | IC50 | 2 | — | |
XFFNHXOXHSUYQQ
|
6.8 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
6.8 | Ki | 66 | — | |
QUCVXIHKWBYLLK
|
6.7 | IC50 | 2 | — | |
OISBNGXKBOCXER
|
6.7 | IC50 | 2 | — | |
TWYKNRDHNFNBDF
|
6.7 | IC50 | 2 | — | |
LKFLRBIQIXBCCO
|
6.7 | IC50 | 2 | — | |
YAVNDOLVFFVVBX
|
6.7 | IC50 | 2 | — | |
AGYZUONRISUOIK
|
6.7 | Ki | 10 | — | |
BLUHZSPELLCJKH
|
6.7 | Ki | 9 | — | |
GCBJDOWIQHMCMR
|
6.7 | Ki | 84 | — | |
HFNKQEVNSGCOJV
|
6.7 | Kd | 65 | — | |
JJJSCYSPSKBQAX
|
6.7 | Ki | 34 | — | |
KNVOICXEDILAGT
|
6.7 | Ki | 17 | — | |
OWDRQHVEJIYVOI
|
6.7 | Ki | 47 | — | |
QRDADMUYUNCQDD
|
6.7 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
6.7 | Ki | 104 | — | |
WPHKIQPVPYJNAX
|
6.7 | Ki | 81 | — | |
YBOOAZFLAUPOKA
|
6.7 | Ki | 3 | — | |
OSVUGUHRKMMBSE
|
6.7 | Kd | 170 | — | |
PQAKQADTDVGYOC
|
6.7 | IC50 | 2 | — |