Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KEBXAEFZLCNLJJ
|
7.1 | Ki | 13 | — | |
RKUKAACYUCUJEE
|
7.1 | Ki | 58 | — | |
VCSQVKQFGYRGEH
|
7.1 | Ki | 13 | — | |
XLFYOIVELARSKP
|
7.1 | Ki | 33 | — | |
YXYNMHMVPRQKBT
|
7.1 | IC50 | 2 | — | |
HZVIUNVVQJWYNZ
|
7.1 | IC50 | 2 | — | |
OJASUOZKOQBQAR
|
7.1 | IC50 | 2 | — | |
QUFSPIHVCCPJER
|
7.1 | IC50 | 2 | — | |
XJFORULEXOZBAQ
|
7.1 | IC50 | 2 | — | |
FWRFPHJSGLYXTD
|
7.1 | IC50 | 3 | — | |
FXMBSEOFWALADX
|
7.0 | IC50 | 3 | — | |
FYKZPCLKTZZIBA
|
7.0 | IC50 | 2 | — | |
VUQPNTNKEPWYRO
|
7.0 | IC50 | 2 | — | |
ALRLENDIHGVVDY
|
7.0 | IC50 | 2 | — | |
VTNHUNPWAHGVCA
|
7.0 | IC50 | 2 | — | |
MCHMLUWPNDLLEY
|
7.0 | IC50 | 2 | — | |
WLLDFEGKGAPLQO
|
7.0 | IC50 | 2 | — | |
ZBKQXBZXZYIRIU
|
7.0 | IC50 | 2 | — | |
DCTBPIBEQFLAOQ
|
7.0 | Ki | 13 | — | |
DFMCXVONDDGQIY
|
7.0 | Ki | 66 | — | |
HEBJJJVAANGHLJ
|
7.0 | IC50 | 2 | — | |
IAKGNUWZPSPEKU
|
7.0 | Ki | 19 | — | |
IJNGXROUMFEKDB
|
7.0 | Ki | 39 | — | |
MCCCQFAOMZMZKE
|
7.0 | Ki | 52 | — | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
YLNVYSOHEOBKJW
|
7.0 | IC50 | 2 | — | |
JSXSJAZHNLZZFG
|
7.0 | IC50 | 2 | — | |
ATCSTBKTLBKJCJ
|
7.0 | Ki | 2 | — | |
FYSLUTGZWHZPCX
|
7.0 | Ki | 2 | — | |
JZBMRMXXSMSEAY
|
7.0 | IC50 | 2 | — | |
OWXKIXPMTVEDCR
|
7.0 | IC50 | 2 | — | |
SQGZUMNITNRRET
|
7.0 | IC50 | 2 | — | |
FXUCGEVPOQUSIH
|
7.0 | IC50 | 2 | — | |
DFAUAZYINZOIAU
|
6.9 | IC50 | 2 | — | |
DUVXFOSLZHSJPX
|
6.9 | Ki | 3 | — | |
SVNVPNHWFJFRLZ
|
6.9 | IC50 | 8 | — | |
GCYXEGSPUDSZJY
|
6.9 | Ki | 82 | — | |
QRCXMLQLNQMAFC
|
6.9 | Ki | 10 | — | |
SQXSMLLCDWJNAC
|
6.9 | Ki | 20 | — | |
XJSFDMGICAWQFS
|
6.9 | Ki | 60 | — | |
XPHWIERLJBFPFV
|
6.9 | Ki | 69 | — | |
XYXLUJQBBIBJFV
|
6.9 | Ki | 36 | — | |
YMIJUBCSOKSFRU
|
6.9 | Ki | 87 | — | |
HKOAGBQDHYMZTP
|
6.9 | IC50 | 2 | — | |
LLDMEDJNOJVTEE
|
6.9 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.9 | Kd | 85 | Yes | |
NHHQJBCNYHBUSI
|
6.9 | Kd | 220 | — | |
NOZFCTAJFMLWPE
|
6.9 | IC50 | 2 | — | |
XEPPZNCGRACPGZ
|
6.9 | IC50 | 2 | — | |
FDYURKPWOPRSMM
|
6.9 | IC50 | 2 | — |