Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FPQBGLUWBCLXFG
|
7.3 | IC50 | 3 | — | |
GCZJQTRRJPRFIP
|
7.3 | Ki | 10 | — | |
HIIXSKLGSBCTAH
|
7.3 | IC50 | 3 | — | |
JVKICFJXJPDNOJ
|
7.3 | IC50 | 2 | — | |
RNFXZZCKTTUGHL
|
7.3 | IC50 | 2 | — | |
LPLVTTVTTDMYHT
|
7.3 | IC50 | 2 | — | |
BMCIBDDLDCNKAP
|
7.3 | IC50 | 2 | — | |
DBLJVNGTXRPKMS
|
7.3 | IC50 | 2 | — | |
FGFUUBCEERIDBQ
|
7.3 | IC50 | 2 | — | |
GAWJEBCHHUPVEO
|
7.3 | IC50 | 2 | — | |
GVYZOWDBQXKJDR
|
7.3 | IC50 | 2 | — | |
HHGUCXDDCLOWPZ
|
7.3 | IC50 | 2 | — | |
IUWQSSGZFYFDEM
|
7.3 | IC50 | 2 | — | |
KLPWXPHBHLDCCS
|
7.3 | IC50 | 2 | — | |
KQXTVRJPONHNFY
|
7.3 | IC50 | 2 | — | |
LXZXQQXBXVENQD
|
7.3 | IC50 | 2 | — | |
MTMFRAIOFPWKIH
|
7.3 | IC50 | 2 | — | |
OLGSXYPPKJJNJR
|
7.3 | IC50 | 2 | — | |
OPZFLEPCEIJFSE
|
7.3 | IC50 | 2 | — | |
PVFRNMLGINKVRT
|
7.3 | IC50 | 2 | — | |
QIMGDBHWVXEGQS
|
7.3 | IC50 | 2 | — | |
RJINHNWMTFJSBN
|
7.3 | IC50 | 2 | — | |
SXKIBLJFZKDDCP
|
7.3 | IC50 | 2 | — | |
UDXGUYCTMQSGOM
|
7.3 | IC50 | 2 | — | |
VMPOUPXTRIFPLU
|
7.3 | IC50 | 2 | — | |
SSHPOTBZTFBVDB
|
7.2 | IC50 | 2 | — | |
UUUBVRVITMLFJU
|
7.2 | IC50 | 2 | — | |
WVIQCXQWRJXXGZ
|
7.2 | IC50 | 2 | — | |
YUDKTFUCCPOVGR
|
7.2 | IC50 | 2 | — | |
QXPNJMHRUZCEAP
|
7.2 | IC50 | 14 | — | |
GHOGNCOJXOPHJS
|
7.2 | IC50 | 2 | — | |
PXYXJSKWHPGJFP
|
7.2 | IC50 | 2 | — | |
SKDBXDGKLQALIZ
|
7.2 | IC50 | 15 | — | |
KWRXWPRFIUJQBP
|
7.2 | Ki | 25 | — | |
QAJPIJHWTGPUNZ
|
7.2 | Ki | 37 | — | |
YJBNTRQKJQHMTM
|
7.2 | Ki | 11 | — | |
ZAYMIFRCEPHPHT
|
7.2 | IC50 | 2 | — | |
HJIRNKSTJOICTI
|
7.2 | IC50 | 2 | — | |
CRQZRBXFLRRAIQ
|
7.2 | Ki | 2 | — | |
RSJWFQUCOMWKQD
|
7.2 | IC50 | 2 | — | |
HXNIAYXLNXQQOW
|
7.2 | IC50 | 2 | — | |
XOAMVMHKXHJDNZ
|
7.2 | IC50 | 2 | — | |
FETVSVYRUZPIRW
|
7.2 | IC50 | 2 | — | |
GVZURVVGRNHCLH
|
7.1 | IC50 | 2 | — | |
SRVMCTQCWVQBNL
|
7.1 | IC50 | 2 | — | |
HMVSRLUUXHNABC
|
7.1 | IC50 | 2 | — | |
IMLMBHVOASBVOW
|
7.1 | IC50 | 2 | — | |
RCCFIMHYOFIWHJ
|
7.1 | IC50 | 2 | — | |
CLEGDJQQHUTCOW
|
7.1 | Ki | 43 | — | |
DKSNLQYRZJKYOC
|
7.1 | Ki | 51 | — |