Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQPLXSNGJYAHSH
|
7.5 | IC50 | 3 | — | |
HVXHSDUKHSDIIZ
|
7.5 | IC50 | 2 | — | |
KVGHGVHKZQAQLD
|
7.5 | IC50 | 3 | — | |
QUVIEDJGNUFDDH
|
7.5 | IC50 | 3 | — | |
SIRSNKXGOCRFCT
|
7.5 | IC50 | 2 | — | |
WSLNKDCNHNOGHL
|
7.5 | IC50 | 3 | — | |
ZJWPYYIRORJZPQ
|
7.5 | IC50 | 4 | — | |
DXBQRCVASKKRRR
|
7.5 | IC50 | 2 | — | |
FKCRUIWBTDNJFG
|
7.5 | IC50 | 4 | — | |
VQBHHVIUAXNAOC
|
7.5 | IC50 | 2 | — | |
PCSNHSCJJFGAOB
|
7.5 | IC50 | 3 | — | |
RRSGLFRYYGSFFX
|
7.5 | IC50 | 2 | — | |
YIHNQOZIZBZUOT
|
7.5 | IC50 | 2 | — | |
CQJWUWZZQUEKGG
|
7.5 | IC50 | 2 | — | |
CMPBIALPWFHSMB
|
7.4 | IC50 | 2 | — | |
GQAOHVZJKCGBQW
|
7.4 | IC50 | 2 | — | |
KGLJXZUKNYLHMK
|
7.4 | IC50 | 2 | — | |
NMGPJZFKRNRWDG
|
7.4 | IC50 | 2 | — | |
PDEDJMZPQFJDNA
|
7.4 | IC50 | 2 | — | |
GEWLYFZWVLXQME
|
7.4 | IC50 | 9 | — | |
VCSAIKGXBLLWTR
|
7.4 | IC50 | 2 | — | |
HWKLPUXMYLCSIE
|
7.4 | IC50 | 2 | — | |
CDELWNRTTCPMLW
|
7.4 | IC50 | 2 | — | |
CLIORPUQKOJRDE
|
7.4 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
7.4 | Ki | 103 | — | |
IOYGZJJCJBOPDM
|
7.4 | Ki | 8 | — | |
PTSMJMBYLZTCHZ
|
7.4 | IC50 | 2 | — | |
UTOQFKLQNHKULZ
|
7.4 | Ki | 2 | — | |
UUQZSFPVUKCRKO
|
7.4 | IC50 | 3 | — | |
CARBAQLLNJEQRM
|
7.4 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
7.4 | IC50 | 2 | — | |
VPJLAZUHVNGPLW
|
7.4 | IC50 | 2 | — | |
FRWDDDSGEGTXIY
|
7.4 | IC50 | 2 | — | |
LFEOCNIHNYNYIJ
|
7.4 | IC50 | 2 | — | |
MOQHPHSZEODHGL
|
7.4 | IC50 | 2 | — | |
DYIZARYDRMKISJ
|
7.4 | IC50 | 2 | — | |
STQNTZGKYOJTGA
|
7.4 | IC50 | 2 | — | |
VFSUAKYNPKYPLY
|
7.4 | Ki | 2 | — | |
KOGDOKSJNXRDBX
|
7.4 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
RVMLNNCKNCFOFH
|
7.4 | IC50 | 4 | — | |
SQBBTXGGRJHRGB
|
7.4 | IC50 | 2 | — | |
LKQCQDSSPGVMPT
|
7.3 | IC50 | 2 | — | |
OWEDOBFUVPKBNA
|
7.3 | IC50 | 2 | — | |
MCHMLUWPNDLLEY
|
7.3 | IC50 | 2 | — | |
AHGFXLZWTGRAAT
|
7.3 | IC50 | 2 | — | |
SHKWWTGWEWLIRC
|
7.3 | IC50 | 2 | — | |
ZAUQVEIJQHLVAR
|
7.3 | IC50 | 2 | — | |
ZDSCMCRGHRMVAM
|
7.3 | IC50 | 2 | — | |
FAYAUAZLLLJJGH
|
7.3 | Ki | 36 | Yes |