Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FEXHRQNJTUVDQQ
|
7.8 | IC50 | 2 | — | |
JONUUBFCZUAOFY
|
7.8 | IC50 | 10 | — | |
RJZDECGDCKOHBV
|
7.8 | Ki | 70 | — | |
UAPCOTPXNOKKFY
|
7.8 | IC50 | 2 | — | |
WTCFYBGLEUOJNE
|
7.8 | IC50 | 2 | — | |
LACOTCUHEDDNGC
|
7.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
QVHDOESZFDSEKS
|
7.7 | Ki | 2 | — | |
RIYDOTWDTHRXAQ
|
7.7 | IC50 | 2 | — | |
ZGXLPGBXVQLLJW
|
7.7 | Ki | 2 | — | |
CSOGCPCCVIPBIK
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | IC50 | 408 | — | |
JYJWZHLMBPNEJV
|
7.7 | IC50 | 2 | — | |
LJNQZRKFYXYCCW
|
7.7 | IC50 | 2 | — | |
XEUHVTVNJONCLA
|
7.7 | IC50 | 2 | — | |
CBAKEHNEEJTUGB
|
7.7 | IC50 | 2 | — | |
NZVDDFRUBIEKLV
|
7.7 | Ki | 20 | — | |
CUBNJCCNGYAEDF
|
7.7 | IC50 | 2 | — | |
CHQYMHAUSYCZKU
|
7.7 | IC50 | 2 | — | |
HUFOBMZPSQAJRA
|
7.7 | IC50 | 2 | — | |
GLKYGVDXWJUOFW
|
7.7 | IC50 | 3 | — | |
IOBRLFTZHXZWPT
|
7.7 | IC50 | 2 | — | |
PFZRXJIYAFANHP
|
7.7 | IC50 | 4 | — | |
CKVWQORGCCEYHS
|
7.6 | Ki | 50 | — | |
FOQNSWUDBARUFL
|
7.6 | IC50 | 3 | — | |
JMHQUQCLIVNTHT
|
7.6 | Ki | 24 | — | |
LRZYYIZFBXFSJB
|
7.6 | Ki | 69 | — | |
NPZBGSCEEAHWNK
|
7.6 | IC50 | 2 | — | |
QONPPIZSNSSCSK
|
7.6 | Ki | 45 | Yes | |
UDRXOUVRNMKWQA
|
7.6 | Ki | 8 | — | |
VUHZDNOPEVGHEO
|
7.6 | Ki | 29 | — | |
TVPNRZPKPMXWJO
|
7.6 | IC50 | 2 | — | |
ACCGDLRUTZSFSS
|
7.6 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
7.6 | IC50 | 2 | — | |
HFTAYZLGTCEXAY
|
7.6 | IC50 | 2 | — | |
JMVDIGHUQAXWIE
|
7.6 | IC50 | 10 | — | |
TVBANCDFRJJEKJ
|
7.6 | IC50 | 2 | — | |
ZIOVJRQVOJIVAE
|
7.6 | IC50 | 2 | — | |
CSOGCPCCVIPBIK
|
7.6 | IC50 | 2 | — | |
OHEKKVOQVJUAQW
|
7.6 | IC50 | 2 | — | |
QKBPOTWGKPRFEH
|
7.6 | IC50 | 2 | — | |
PEHQJHHHTXOGJK
|
7.6 | IC50 | 2 | — | |
QHADVLVFMKEIIP
|
7.6 | IC50 | 9 | — | |
DGUSKGFGXIHXKS
|
7.5 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
7.5 | IC50 | 2 | — | |
ILYKJXYOFZKJGR
|
7.5 | IC50 | 2 | — | |
LEAJNJJPWHYFJT
|
7.5 | IC50 | 2 | — | |
KAZFNRNYKKXSJQ
|
7.5 | IC50 | 2 | — | |
CQPDKJQEKIKEFC
|
7.5 | IC50 | 2 | — | |
DPFZKILBVWKIDP
|
7.5 | IC50 | 3 | — |