Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FMGALEFRCKPSHT
|
8.2 | IC50 | 2 | — | |
MPUZHXLKCBEGNC
|
8.2 | IC50 | 2 | — | |
OJGVXOPNHCRTAD
|
8.2 | IC50 | 2 | — | |
DUHHTOOYELYHTE
|
8.2 | IC50 | 2 | — | |
RKNGTCDEHZFRSK
|
8.2 | IC50 | 2 | — | |
FWTKVRZMQJINSD
|
8.2 | IC50 | 5 | — | |
GXGBEOFIFZVLQU
|
8.2 | IC50 | 2 | — | |
BIBRQIOPTKIPOZ
|
8.1 | IC50 | 2 | — | |
PYMYZZLESAPEGL
|
8.1 | IC50 | 2 | — | |
VENBOQULCZPZRI
|
8.1 | IC50 | 2 | — | |
ZMKWRVSEWQLUIX
|
8.1 | IC50 | 2 | — | |
CXNIDEGZWPEOCF
|
8.1 | IC50 | 3 | — | |
DXRIPNKUBZNZQN
|
8.1 | IC50 | 2 | — | |
FCCJIRJUDAWXRO
|
8.1 | IC50 | 4 | — | |
KKBIMZUEOUDERI
|
8.1 | IC50 | 2 | — | |
UKTICNMOUVEYRR
|
8.1 | IC50 | 4 | — | |
ZDNCMUXDGZVSHU
|
8.1 | IC50 | 2 | — | |
MOHKECCWMOAJNH
|
8.1 | IC50 | 2 | — | |
DTEWSDGBCMIPIZ
|
8.1 | IC50 | 2 | — | |
CJQYSYNGPPQQJW
|
8.1 | IC50 | 2 | — | |
QZAPGJZGBUIRLB
|
8.1 | IC50 | 2 | — | |
VCRXHIDEBJOEFB
|
8.1 | IC50 | 2 | — | |
HNWUOUYCKCPSHE
|
8.1 | IC50 | 2 | — | |
NFYSHFWLDDXPKM
|
8.1 | IC50 | 3 | — | |
QSNAMJCLIIQNPP
|
8.1 | IC50 | 2 | — | |
BFUCQUQBTJOBTA
|
8.0 | IC50 | 3 | — | |
DCUJQHLLVMQMID
|
8.0 | IC50 | 2 | — | |
MCHMLUWPNDLLEY
|
8.0 | IC50 | 2 | — | |
VFWWHCOMWRSXME
|
8.0 | IC50 | 2 | — | |
CGMQSJXTBXHOTH
|
8.0 | IC50 | 9 | — | |
LXOPXNJLPKCVBS
|
8.0 | IC50 | 2 | — | |
LZDLAOSZVOKASQ
|
8.0 | IC50 | 2 | — | |
XOJQJDHWKVZUAT
|
8.0 | Ki | 9 | — | |
PXKYYYJETYKSIZ
|
8.0 | IC50 | 2 | — | |
OVAFHXUOPSXQOF
|
8.0 | IC50 | 2 | — | |
GEWLYFZWVLXQME
|
8.0 | IC50 | 2 | — | |
GUXLMYYFWLSMCP
|
8.0 | IC50 | 2 | — | |
KTBKRHUBYKAUFQ
|
8.0 | IC50 | 2 | — | |
MLNZVQPAJITTGP
|
8.0 | IC50 | 2 | — | |
SIILILXNZLEIIT
|
8.0 | IC50 | 2 | — | |
ANUKWIYBPKFKPT
|
7.9 | IC50 | 2 | — | |
IXQFWQXAZJXVSH
|
7.9 | IC50 | 2 | — | |
KXZLWAAQYGMLJX
|
7.9 | IC50 | 3 | — | |
PJFYYYJFEHNOHR
|
7.9 | IC50 | 2 | — | |
AJGPWESAFONVCG
|
7.9 | IC50 | 3 | — | |
HHFBDROWDBDFBR
|
7.9 | IC50 | 40 | Yes | |
UXNUQVZRIJPJBL
|
7.8 | IC50 | 2 | — | |
VQZTVBGPAZGVHT
|
7.8 | IC50 | 2 | — | |
OGNWKFYJHNZTNC
|
7.8 | IC50 | 2 | — | |
DJPQIFRWWIYXCH
|
7.8 | IC50 | 2 | — |