Target Details
| UniProt AC | Q9HBH9 |
|---|---|
| Gene Symbol | MKNK2 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 608
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (3)
Active Molecules (608)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JEOHNIZYSBQLBI
|
9.9 | IC50 | 2 | — | |
XRIMGCCVXQKXAF
|
9.8 | IC50 | 2 | — | |
GBZIOQYCTAFXKL
|
9.4 | IC50 | 2 | — | |
HDKZJMGFRSXWSJ
|
9.4 | IC50 | 3 | — | |
ZRIDICSQDPQVEH
|
9.3 | IC50 | 3 | — | |
GXUYZVYTXZYDQM
|
9.2 | IC50 | 3 | — | |
CDWDPWNPTCKJNW
|
9.2 | IC50 | 2 | — | |
XCYFTLJVXBVKHG
|
9.2 | IC50 | 2 | — | |
DHFSWODVDVUGGC
|
9.2 | IC50 | 3 | — | |
WCADNSJQHAGKBX
|
9.2 | IC50 | 3 | — | |
CYVKSJTVMXLBEL
|
9.1 | IC50 | 2 | — | |
CUSAZOGXBMLNCR
|
9.0 | IC50 | 2 | — | |
DZCGBMMTMNQQHW
|
9.0 | IC50 | 2 | — | |
GCMXEMBFFWKSQR
|
9.0 | IC50 | 2 | — | |
GKGFTCRWDLEQNT
|
9.0 | IC50 | 2 | — | |
IHHXSJUBRJFSFB
|
9.0 | IC50 | 2 | — | |
JONIGSIXPCHLPF
|
9.0 | IC50 | 3 | — | |
KBJGQQRVHPTDJO
|
9.0 | IC50 | 2 | — | |
LGXIHGFTIXRTGJ
|
9.0 | IC50 | 2 | — | |
OYOKXIIAQLUGEQ
|
9.0 | IC50 | 2 | — | |
PNJVSKGBROJKNX
|
9.0 | IC50 | 2 | — | |
QCKSDSPCHDSAHA
|
9.0 | IC50 | 2 | — | |
SHFKCVNKUAWFOE
|
9.0 | IC50 | 2 | — | |
TXTSSJDYULDSBL
|
9.0 | IC50 | 2 | — | |
VKZOMKUUMGEJLL
|
9.0 | IC50 | 2 | — | |
WSPFOBDEROUNMO
|
9.0 | IC50 | 2 | — | |
XCQQKYFEUUGRAR
|
9.0 | IC50 | 2 | — | |
YCHQXPNHRHYUIG
|
9.0 | IC50 | 2 | — | |
YFJVDNQENDFYRT
|
9.0 | IC50 | 2 | — | |
HKTBYUWLRDZAJK
|
9.0 | IC50 | 5 | — | |
YRDRYCRFGSQZQW
|
9.0 | IC50 | 2 | — | |
POSZZZFFLNLQCL
|
8.9 | IC50 | 3 | — | |
RZKFMYXHNVBJJV
|
8.9 | IC50 | 2 | — | |
VPIDNMQLFOKKCY
|
8.9 | IC50 | 2 | — | |
ZZONCZDKYUYGTE
|
8.9 | IC50 | 2 | — | |
JMOODDNVNBVCOJ
|
8.9 | IC50 | 3 | — | |
NTLQCWXRQTUIRI
|
8.9 | IC50 | 2 | — | |
PFYNAVHEBIAEKL
|
8.9 | IC50 | 2 | — | |
FOGVEYPAPSELLE
|
8.8 | IC50 | 2 | — | |
FWTDZBZYPAAGCF
|
8.8 | IC50 | 2 | — | |
IPJHWPFFKVRFPR
|
8.8 | IC50 | 2 | — | |
MNORXFRHDOWTKB
|
8.8 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.8 | Kd | 289 | Yes | |
LCQIIAREQLPINL
|
8.8 | IC50 | 2 | — | |
LGDROMVQTALVNT
|
8.8 | IC50 | 3 | — | |
RWDCJKPJKMBFCI
|
8.8 | IC50 | 2 | — | |
WCADNSJQHAGKBX
|
8.8 | IC50 | 3 | — | |
RBEFDXXUUNMTSK
|
8.8 | IC50 | 2 | — | |
UXHZMEYLBGGTQR
|
8.8 | IC50 | 2 | — | |
VQBHHVIUAXNAOC
|
8.8 | IC50 | 3 | — |