Target Details
| UniProt AC | Q9HB55 |
|---|---|
| Gene Symbol | CYP3A43 |
| Protein Name | Cytochrome P450 3A43 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00067 (p450) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DOLFOQBBXQXIND
|
8.9 | Ki | 4 | — | |
LJVAJPDWBABPEJ
|
8.6 | Ki | 59 | — | |
WQQQUDROKZMYJS
|
8.3 | Ki | 4 | — | |
FDQOBNRCVYTPOK
|
8.2 | Ki | 4 | — | |
IMZNBJHINVKCOT
|
7.6 | Ki | 4 | — | |
KNDXCMQNZXPRGV
|
7.6 | Ki | 4 | — | |
NCDNCNXCDXHOMX
|
7.4 | IC50 | 12 | — | |
WDWIMDKOXZZYHH
|
6.6 | IC50 | 4 | — | |
GXMINRJZNGLAOL
|
6.6 | IC50 | 29 | — | |
BLMPQMFVWMYDKT
|
6.3 | IC50 | 43 | — | |
XMTPWAPSQQBCQF
|
6.2 | IC50 | 4 | — | |
BCEHBSKCWLPMDN
|
6.2 | Ki | 10 | — | |
QJJXYPPXXYFBGM
|
6.2 | IC50 | 11 | — | |
JAHXQCZCZURPTI
|
6.2 | IC50 | 34 | — | |
JBZRAEUHDPMQSF
|
6.0 | IC50 | 34 | — | |
PMATZTZNYRCHOR
|
6.0 | Ki | 20 | — |