Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVUWQDLBEOZVOU
|
7.8 | IC50 | 41 | — | |
YKFHBMIPXGSMRS
|
7.8 | IC50 | 7 | — | |
YRFAWSIUIFNVQA
|
7.8 | IC50 | 9 | — | |
YSBCFQVEEKUZSU
|
7.8 | IC50 | 7 | — | |
CXJCGSPAPOTTSF
|
7.8 | IC50 | 6 | — | |
ANKYADWZYKSCAJ
|
7.8 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
JQHTYMOOIFVIJV
|
7.8 | IC50 | 5 | — | |
KOZFSFOOLUUIGY
|
7.8 | Kd | 88 | Yes | |
MEZZCEDCBNWCRR
|
7.8 | IC50 | 7 | — | |
QKCAXXVNZDAJAD
|
7.8 | IC50 | 5 | — | |
RUQXGVGYNKIGJD
|
7.8 | IC50 | 7 | — | |
BQYDGSNDLAZAEW
|
7.8 | Ki | 13 | — | |
GWXPHWSUMLUDPO
|
7.8 | Ki | 11 | — | |
IRBWROIEALHOPH
|
7.8 | IC50 | 7 | — | |
PCQMERRARZKTPW
|
7.8 | Ki | 68 | — | |
RPGBQFNDFPEOON
|
7.8 | Ki | 22 | — | |
SZALFSTUDMTGGL
|
7.8 | Ki | 3 | — | |
UJBJWYNPUOLFIZ
|
7.8 | Ki | 49 | — | |
UYJNQQDJUOUFQJ
|
7.8 | Ki | 68 | — | |
VBIYDORVDCFKHM
|
7.8 | Ki | 13 | — | |
WQYUNADCLFWKGN
|
7.8 | IC50 | 7 | — | |
WYLVFMBGPRCDQF
|
7.8 | Ki | 14 | — | |
XTJRKTBELWGSDN
|
7.8 | IC50 | 8 | — | |
GUXARCGBVPDGMI
|
7.8 | IC50 | 3 | — | |
QHTJZFWEQYRYQE
|
7.8 | IC50 | 9 | — | |
AAYFHKFUAWLHMY
|
7.8 | IC50 | 5 | — | |
OEVQTWCGWDOIFZ
|
7.8 | IC50 | 7 | — | |
XQQYRDDJENLAME
|
7.8 | IC50 | 8 | — | |
ANKYADWZYKSCAJ
|
7.8 | IC50 | 7 | — | |
OWDVXJJCVWTPPW
|
7.8 | IC50 | 8 | — | |
PPALZSWDMRGSQV
|
7.8 | IC50 | 5 | — | |
WROAXSSJZFFCSV
|
7.7 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.7 | Kd | 165 | Yes | |
CHQYAWLKOUOTQO
|
7.7 | IC50 | 7 | — | |
NVTNPVQFMSQPJQ
|
7.7 | IC50 | 7 | — | |
QDNBLKZVYODRLC
|
7.7 | IC50 | 5 | — | |
UGYUFJPHSWYELP
|
7.7 | IC50 | 8 | — | |
AHJRHEGDXFFMBM
|
7.7 | Ki | 28 | — | |
CLRFYTGANQZOBS
|
7.7 | Ki | 41 | — | |
FAIHBCXQSBIRIL
|
7.7 | Ki | 22 | — | |
GHAZVJQMLWOQLP
|
7.7 | Ki | 17 | — | |
JEPGNFQKCRZPHJ
|
7.7 | IC50 | 3 | — | |
MCKPYPWHBUXLEZ
|
7.7 | Ki | 21 | — | |
OUJZYQBEFNDJQN
|
7.7 | Ki | 71 | — | |
PAEFKCSDRFLRMD
|
7.7 | IC50 | 5 | — | |
RRAMBEGOYIJQHY
|
7.7 | Ki | 11 | — | |
WHVFDYQCAMPLMS
|
7.7 | Ki | 20 | Yes | |
XYFHSCKRPLMJIO
|
7.7 | IC50 | 3 | — | |
YJBNTRQKJQHMTM
|
7.7 | Ki | 11 | — |