Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CBTNARFZVOPLBO
|
8.0 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
8.0 | IC50 | 7 | — | |
GCSZJMUFYOAHFY
|
8.0 | IC50 | 8 | — | |
IJFKKIMDRSZOOW
|
8.0 | IC50 | 6 | — | |
MUOKSQABCJCOPU
|
8.0 | IC50 | 36 | — | |
QNWARURWFRZNNO
|
8.0 | IC50 | 7 | — | |
RAQBQAXSLHDSKW
|
8.0 | IC50 | 8 | — | |
SBYPANVVFZBWDF
|
8.0 | IC50 | 9 | — | |
YAXGFAAKCUOWNM
|
8.0 | IC50 | 9 | — | |
VCCCOYOXNKTQFO
|
7.9 | IC50 | 9 | — | |
YGVKOSRPXIWQPQ
|
7.9 | IC50 | 4 | — | |
CRVHQVJVMWGKAV
|
7.9 | IC50 | 3 | — | |
HEAGNKNMQVIVMM
|
7.9 | IC50 | 8 | — | |
HHSNDNONCUTNQR
|
7.9 | IC50 | 7 | — | |
IDOKKOQIQLHASZ
|
7.9 | IC50 | 8 | — | |
JTYIDARLAQQHPP
|
7.9 | IC50 | 4 | — | |
LXDHFJUOCGKVAV
|
7.9 | IC50 | 5 | — | |
MJXIIYIGVBRQNO
|
7.9 | IC50 | 4 | — | |
MXEZQEFCKXVMFN
|
7.9 | IC50 | 5 | — | |
QCHDHJOEPUQALZ
|
7.9 | IC50 | 9 | — | |
QVYXLOYBJBMXNP
|
7.9 | IC50 | 7 | — | |
VJSOYRZFTRFBFM
|
7.9 | IC50 | 5 | — | |
AOBLBPWPSKBHSI
|
7.9 | Ki | 55 | — | |
CPGKMMMSMJKHDL
|
7.9 | Ki | 16 | — | |
FLEAYYMORDPWAJ
|
7.9 | Ki | 90 | — | |
FQEODTMNWMDUMD
|
7.9 | Ki | 25 | — | |
GCBJDOWIQHMCMR
|
7.9 | Ki | 84 | — | |
HZGYSSZTTMUCJE
|
7.9 | Ki | 8 | — | |
IUEBPIPDFMCSTP
|
7.9 | Ki | 29 | — | |
JLTBOCSFMNSLFH
|
7.9 | Ki | 9 | — | |
OQHALFBQFMAXFZ
|
7.9 | Ki | 9 | — | |
QRCXMLQLNQMAFC
|
7.9 | Ki | 10 | — | |
RQJIDUOCLNMUHR
|
7.9 | Ki | 15 | — | |
VVEGARMQKNYDID
|
7.9 | Ki | 24 | — | |
ACOQCSBMVFAWQV
|
7.9 | IC50 | 8 | — | |
AYCPARAPKDAOEN
|
7.9 | Kd | 73 | — | |
KQCIEIGKPXQRLM
|
7.9 | IC50 | 6 | — | |
KQZBWTMAFLOSPA
|
7.9 | IC50 | 8 | — | |
URXJBXVGNBGIJA
|
7.9 | IC50 | 9 | — | |
XCTYEZWILVGTGO
|
7.9 | IC50 | 9 | — | |
PBVAHEBIEXXNNA
|
7.9 | IC50 | 4 | — | |
ZDJFIKFQLKJRBA
|
7.9 | IC50 | 4 | — | |
FFJGYBJUQCZAAY
|
7.8 | IC50 | 5 | — | |
GXCOUFPTCZUTEE
|
7.8 | IC50 | 10 | — | |
HAFFBDGNUZMNIJ
|
7.8 | IC50 | 7 | — | |
IDGNCVHQDDOPND
|
7.8 | IC50 | 6 | — | |
JNTIINGGIOJIMW
|
7.8 | IC50 | 4 | — | |
JXQZHHAAJMQJKU
|
7.8 | IC50 | 6 | — | |
KBEZZFIQPRMPRG
|
7.8 | IC50 | 5 | — | |
RVYFLJXKEYHVBR
|
7.8 | IC50 | 5 | — |