Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AWDORCFLUJZUQS
|
6.0 | Ki | 22 | — | |
BHDRCBRVTBITOC
|
6.0 | IC50 | 2 | — | |
BMKHCMLGQGVJTF
|
6.0 | Ki | 2 | — | |
BNLPAUPVSCPTDM
|
6.0 | Ki | 15 | — | |
GMYYMEOGFRKSFS
|
6.0 | Ki | 29 | — | |
GTMGQYXCPKUZAD
|
6.0 | Ki | 6 | Yes | |
HOBMVEVXDIOMDM
|
6.0 | Ki | 18 | — | |
ITAJXWHXKVYGCF
|
6.0 | Ki | 5 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KWSZYBNXNYRQCC
|
6.0 | Ki | 21 | — | |
LCYPRFCDTJTQPG
|
6.0 | Ki | 5 | — | |
LHNIIDJUOCFXAP
|
6.0 | Ki | 20 | Yes | |
LRINYHMQZRENCY
|
6.0 | Ki | 29 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MTSNDBYBIZSILH
|
6.0 | Ki | 2 | — | |
NPLQZQGAZAUUTB
|
6.0 | Ki | 9 | — | |
NWAUBAGBGOPJLF
|
6.0 | Ki | 51 | Yes | |
OULGHWYAFYSZGK
|
6.0 | Ki | 2 | — | |
PBBRWFOVCUAONR
|
6.0 | Ki | 26 | Yes | |
RPGMSHCJIWHISY
|
6.0 | IC50 | 3 | — | |
RPGMSHCJIWHISY
|
6.0 | IC50 | 3 | — | |
RTYJMUXLFRYRBU
|
6.0 | Ki | 35 | — | |
SJDGHXXYFFXVPE
|
6.0 | Ki | 9 | — | |
UNVKXVCDLOLPJE
|
6.0 | Ki | 8 | — | |
UOVCGJXDGOGOCZ
|
6.0 | Ki | 59 | — | |
VSPFURGQAYMVAN
|
6.0 | Ki | 17 | — | |
WPHKIQPVPYJNAX
|
6.0 | Ki | 81 | — | |
YRVHWCZERXVDLL
|
6.0 | Ki | 6 | — | |
ZNOLRTPMNMPLHY
|
6.0 | Kd | 6 | — |