Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QKPLUKMJEKRAJD
|
6.3 | Ki | 30 | Yes | |
RIUZPIBUSOHUKF
|
6.3 | Ki | 23 | — | |
ROPVGAMDOWWUTK
|
6.3 | Ki | 5 | — | |
SDTHQOXRWZXTJF
|
6.3 | Ki | 16 | — | |
UMYBAQLXZPEUQW
|
6.3 | Ki | 15 | — | |
UTBSBSOBZHXMHI
|
6.3 | IC50 | 3 | — | |
VRIFJAKXSBXYFZ
|
6.3 | Ki | 8 | — | |
WVFWTUJEHMVUBG
|
6.3 | Ki | 25 | — | |
XFUXPAURFGNBSI
|
6.3 | Ki | 4 | — | |
YKYRQCWLYUTVIE
|
6.3 | Ki | 16 | — | |
YYPKOMNJRZRWIC
|
6.3 | Ki | 26 | — | |
YZHOOLPUTYUPEQ
|
6.3 | Ki | 2 | — | |
ZKHDDJKHTPLPOQ
|
6.3 | Ki | 62 | — | |
JDUBGYFRJFOXQC
|
6.3 | Kd | 13 | — | |
PBGPFWACZLCJFH
|
6.3 | IC50 | 3 | — | |
SEERTRJTWMFXIC
|
6.3 | IC50 | 2 | — | |
BAUOZGQJLRLMNO
|
6.2 | IC50 | 4 | — | |
HDBIRBUHIXXLDF
|
6.2 | IC50 | 4 | — | |
BTIHMVBBUGXLCJ
|
6.2 | IC50 | 21 | Yes | |
YCFRZMCRPHNZOC
|
6.2 | IC50 | 7 | — | |
YCFRZMCRPHNZOC
|
6.2 | IC50 | 6 | — | |
AOFJRBMLTUGMMP
|
6.2 | Ki | 12 | — | |
CACMTVGXYAZZNY
|
6.2 | Ki | 11 | — | |
CKVWQORGCCEYHS
|
6.2 | Ki | 50 | — | |
DKSNLQYRZJKYOC
|
6.2 | Ki | 51 | — | |
FAYAUAZLLLJJGH
|
6.2 | Ki | 36 | Yes | |
GNZPMJDEUIVORU
|
6.2 | Ki | 3 | — | |
HRJWTAWVFDCTGO
|
6.2 | Ki | 13 | Yes | |
IJRBJCMLWLFMIN
|
6.2 | Ki | 17 | — | |
JIFGOPCFXJIPNK
|
6.2 | Ki | 5 | — | |
JPJBCKSRGYPABG
|
6.2 | IC50 | 3 | — | |
LWBSSNRDDDFHSH
|
6.2 | Ki | 9 | — | |
NPHKXSDZIKFIRU
|
6.2 | Ki | 5 | — | |
OBHNPUMYQHGYJJ
|
6.2 | Ki | 4 | — | |
OMKZJNFKGWJFNX
|
6.2 | Ki | 8 | — | |
OQSVYNYDHYYKJX
|
6.2 | Ki | 7 | — | |
QCOULMVHIHJKFY
|
6.2 | Ki | 14 | — | |
QNZJDYVERIAXAI
|
6.2 | Ki | 7 | — | |
QXRJBJVCBQSLTA
|
6.2 | Ki | 29 | — | |
SYSUZXPGQXEWCZ
|
6.2 | Ki | 10 | — | |
VUHZDNOPEVGHEO
|
6.2 | Ki | 29 | — | |
XIOOJUQFJYPVLA
|
6.2 | Ki | 17 | — | |
XTVULKIROSNNTG
|
6.2 | Ki | 29 | — | |
YGEACCLUBSGMMJ
|
6.2 | Ki | 16 | — | |
YOVNFNXUCOWYSG
|
6.2 | Ki | 33 | Yes | |
ZVPDNRVYHLRXLX
|
6.2 | Ki | 35 | Yes | |
HFZLFYUNSURMIG
|
6.2 | IC50 | 3 | — | |
ZYDSDRZMIWGATN
|
6.2 | IC50 | 3 | — | |
IXTKPNOXAVTBCW
|
6.2 | IC50 | 4 | — | |
NPCHLCRENQCWNN
|
6.2 | IC50 | 2 | — |