Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — | |
YRFAWSIUIFNVQA
|
7.0 | IC50 | 4 | — | |
DLDXMINZRQNSDI
|
7.0 | IC50 | 3 | — | |
HMDPCTZKMDHQTP
|
7.0 | IC50 | 5 | — | |
TYCNIAHUXCRTIA
|
7.0 | IC50 | 2 | — | |
GIQDYWGEMOCDSN
|
7.0 | IC50 | 5 | — | |
RDXUXJLQXOFAJG
|
7.0 | IC50 | 4 | — | |
UTBSBSOBZHXMHI
|
7.0 | IC50 | 15 | Yes | |
VDJFUWZMISVQGO
|
7.0 | IC50 | 4 | — | |
GQBQUBULFDQKBM
|
7.0 | IC50 | 4 | — | |
QQWUGDVOUVUTOY
|
7.0 | Kd | 231 | Yes | |
RPGZQOOZHIEPJW
|
7.0 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.0 | Kd | 18 | — | |
TZFBRBFUNGMUNQ
|
7.0 | IC50 | 3 | — | |
COYCDCAUDJBGOV
|
7.0 | IC50 | 6 | — | |
BWUOLNXJAQPJKF
|
6.9 | IC50 | 7 | — | |
MCUJGJCMGRDTIE
|
6.9 | IC50 | 2 | — | |
NDCWSHMFDBDIQV
|
6.9 | IC50 | 3 | — | |
CYVGSDYVNUNREA
|
6.9 | IC50 | 5 | — | |
DKKAPUBGRWMMGK
|
6.9 | IC50 | 5 | — | |
LASLZTNNTZVYMJ
|
6.9 | IC50 | 4 | — | |
VCZRYZZCLOMGOV
|
6.9 | IC50 | 4 | — | |
ZYDSDRZMIWGATN
|
6.9 | IC50 | 3 | — | |
CNCRCDLWUGCPSJ
|
6.9 | IC50 | 5 | — | |
CYUDBMRFRZUOTH
|
6.9 | IC50 | 5 | — | |
DZSUJUOJJJCWGG
|
6.9 | Ki | 55 | Yes | |
FANUXQYVRUHAAH
|
6.9 | IC50 | 6 | — | |
FPLAQCFCGCSDRB
|
6.9 | Ki | 4 | — | |
GHMRUNOHAHJNNA
|
6.9 | Ki | 29 | — | |
GLMWKEAUVZDGKE
|
6.9 | Ki | 23 | — | |
HHSVICUMCOBRPT
|
6.9 | Ki | 33 | — | |
KYACBMRLQMEIAI
|
6.9 | Ki | 30 | — | |
LDNVJIDFNXGSGT
|
6.9 | IC50 | 6 | — | |
MHWHPWMWKYXCRJ
|
6.9 | Ki | 32 | — | |
MLGGUGPIWDHBAI
|
6.9 | IC50 | 10 | — | |
MLGGUGPIWDHBAI
|
6.9 | Ki | 33 | — | |
NEWAULHLLUCDPD
|
6.9 | Ki | 27 | — | |
NMHMCXTYPRADBA
|
6.9 | Ki | 20 | — | |
NRSGWEVTVGZDFC
|
6.9 | Ki | 50 | — | |
PNKALLUVKOKYHZ
|
6.9 | Ki | 32 | — | |
WZISGNDZZPSYRP
|
6.9 | Ki | 20 | — | |
XGMWRIIMIJPGBH
|
6.9 | Ki | 10 | — | |
XLFYOIVELARSKP
|
6.9 | Ki | 33 | — | |
YGKFZWJWKPZPQM
|
6.9 | Ki | 13 | — | |
ZCBUQCWBWNUWSU
|
6.9 | Ki | 11 | — | |
MYVQRBFVXBKGNN
|
6.9 | IC50 | 2 | — | |
UFGCTWUIESUHQP
|
6.9 | IC50 | 7 | — | |
UJIAQDJKSXQLIT
|
6.9 | Kd | 38 | — | |
FVIUKIZPDJZQKD
|
6.9 | IC50 | 5 | — | |
GFOASKPCKCZBDL
|
6.9 | IC50 | 2 | — |