Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTHYGYNOCOBONC
|
7.3 | IC50 | 4 | — | |
PAHHKMMVQJCPJI
|
7.2 | IC50 | 8 | — | |
QSGKPYRFWJINEH
|
7.2 | IC50 | 12 | — | |
ZHTZVZJNJGCSJO
|
7.2 | IC50 | 7 | — | |
HZTYDQRUAWIZRE
|
7.2 | Kd | 40 | Yes | |
CSNGPDJYNPSXNA
|
7.2 | IC50 | 5 | — | |
DLDXMINZRQNSDI
|
7.2 | IC50 | 3 | — | |
IFLBFWBMAWIBBZ
|
7.2 | Kd | 7 | — | |
BLUHZSPELLCJKH
|
7.2 | Ki | 9 | — | |
HDEZJSLYUKYKAZ
|
7.2 | Ki | 6 | — | |
IPTSYCYNQJITNJ
|
7.2 | Ki | 12 | — | |
JBLPUDJLELBRHC
|
7.2 | Ki | 9 | — | |
KBDRSPRFXNCQAM
|
7.2 | Ki | 8 | — | |
KIEFRRZUZZNWHT
|
7.2 | Ki | 6 | — | |
KIUHBHFVVQQALF
|
7.2 | Ki | 9 | — | |
KNACLJBHKVSTDL
|
7.2 | Ki | 40 | — | |
LACOMQAWPSFXQC
|
7.2 | Ki | 27 | — | |
MZDKLVOWGIOKTN
|
7.2 | Ki | 80 | — | |
OEEGUWWPGAZRIJ
|
7.2 | Ki | 21 | — | |
OWFLADWRSCINST
|
7.2 | Ki | 30 | — | |
PHWHNHYZZNJPLB
|
7.2 | Ki | 16 | — | |
SHENEEFOURUIBP
|
7.2 | Ki | 29 | — | |
UXUQVXDYXKMCGA
|
7.2 | Ki | 21 | — | |
VAMDLIMJLAPZGX
|
7.2 | Ki | 10 | — | |
WRZNQKSBJJKEBD
|
7.2 | Ki | 6 | — | |
XOVPCPRZRHQFBI
|
7.2 | Ki | 15 | — | |
YGUMGYOBTNGZKS
|
7.2 | Ki | 12 | — | |
ZYFRJAWGLQYBTJ
|
7.2 | IC50 | 5 | — | |
ADJWQFUAOONPHD
|
7.2 | IC50 | 8 | — | |
UMYSGMXAOXMMGG
|
7.2 | IC50 | 7 | — | |
GJYVLTPTDBQQCY
|
7.2 | IC50 | 7 | — | |
JQSJAVBMIMDUFO
|
7.2 | IC50 | 4 | — | |
JPJBCKSRGYPABG
|
7.2 | IC50 | 3 | — | |
OSWHZHVVVZAPRN
|
7.2 | IC50 | 6 | — | |
AQDWDWAYVBQMAM
|
7.2 | IC50 | 7 | — | |
NJETXHOGHMMTEB
|
7.2 | IC50 | 4 | — | |
NRHKUKQUEJSGMG
|
7.2 | IC50 | 3 | — | |
PGPHHJBZEGSUNE
|
7.2 | Kd | 17 | — | |
RUQXGVGYNKIGJD
|
7.2 | IC50 | 4 | — | |
VNRLVGZOAVIXDU
|
7.2 | IC50 | 4 | — | |
FFESRGFMLQEDRD
|
7.1 | IC50 | 5 | — | |
WYVDFOFDVCFARJ
|
7.1 | IC50 | 6 | — | |
GPXCDUCDIFDAGL
|
7.1 | IC50 | 3 | — | |
JGJABYQWCCWLPP
|
7.1 | IC50 | 4 | — | |
MXIKVRCYCKFUND
|
7.1 | IC50 | 6 | — | |
BQWUBCRDJPIJAT
|
7.1 | Ki | 10 | — | |
BUDGLAJKNWCXIM
|
7.1 | IC50 | 4 | — | |
CTJAMSGCMYAVCZ
|
7.1 | Ki | 14 | — | |
CZIGMBNEFWBEMD
|
7.1 | Ki | 16 | — | |
DBKQWGCVGCVPIP
|
7.1 | Ki | 21 | — |