Target Details
| UniProt AC | Q9HAZ1 |
|---|---|
| Gene Symbol | CLK4 |
| Protein Name | Dual specificity protein kinase CLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 930
- Clinical molecules 37
- Avg pChEMBL 7.25
KEGG Pathways (1)
Active Molecules (930)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWMPVMMGSHXANZ
|
9.5 | Ki | 58 | — | |
BPNUQXPIQBZCMR
|
9.3 | Kd | 83 | Yes | |
PMWVYONICYRLNY
|
9.2 | Kd | 4 | — | |
RKUKAACYUCUJEE
|
9.2 | Ki | 58 | — | |
URNZTLZSAVLTIZ
|
9.2 | Ki | 26 | — | |
KYOPCGIPHGGWMV
|
9.1 | Kd | 7 | — | |
BBCSUMURJUYILA
|
9.0 | IC50 | 10 | — | |
BQWWOBKMDWACGC
|
9.0 | IC50 | 8 | — | |
HZPACYSNLOCDLW
|
9.0 | Ki | 48 | — | |
JFDRONLMXPRQPP
|
9.0 | IC50 | 9 | — | |
LHQWPYOYDRVMFI
|
9.0 | Ki | 21 | — | |
WDARYLSSWBWVCU
|
9.0 | Ki | 49 | — | |
YSODDCRKIDDXKM
|
9.0 | IC50 | 9 | — | |
BEJCLDKQCNVTQR
|
8.9 | Ki | 16 | — | |
BGYVWFZMYBWCNY
|
8.9 | Ki | 30 | — | |
ACSYKUPGCXYRRO
|
8.8 | Ki | 26 | — | |
BWNQBFHVFFZHMR
|
8.7 | IC50 | 10 | — | |
CNQGNADBGYCKKV
|
8.7 | Ki | 25 | — | |
DPDVVGCNUWGGRS
|
8.7 | IC50 | 10 | — | |
DXVSNYWBRDTHFF
|
8.7 | IC50 | 10 | — | |
HKSZLNNOFSGOKW
|
8.7 | Ki | 118 | — | |
HXESDBWWDYJEJQ
|
8.7 | Ki | 10 | — | |
IEFFSHLHNYVSEF
|
8.7 | IC50 | 8 | — | |
NBTJWRPKGNQBJS
|
8.7 | IC50 | 8 | — | |
QMUKOEKTUBVPFU
|
8.7 | IC50 | 12 | — | |
QXFBTYPBHYOEMX
|
8.7 | IC50 | 9 | — | |
RJYLSCSDDDQEPD
|
8.7 | IC50 | 10 | — | |
SLKCVFPEQGHNSI
|
8.7 | Ki | 29 | — | |
XLSYZSRXVVCHLS
|
8.7 | Kd | 48 | — | |
YEZMGVBTPDYRPO
|
8.7 | IC50 | 8 | — | |
DPIAIAIQEINUNP
|
8.7 | IC50 | 4 | — | |
HHUOQHKKRABAQB
|
8.6 | IC50 | 5 | — | |
JJTYLBBKGQOISV
|
8.6 | Ki | 15 | — | |
XUFLBSMTYMFOQH
|
8.6 | Ki | 43 | — | |
FSBMCTDYWXIBLM
|
8.6 | IC50 | 22 | — | |
YRFOQHHFWYWAST
|
8.5 | IC50 | 22 | — | |
BUDHVVXPBGMAPV
|
8.5 | IC50 | 11 | — | |
BULHRWBHKAVJMT
|
8.5 | IC50 | 8 | — | |
CGPYAXSYKQBYKJ
|
8.5 | IC50 | 12 | — | |
FIVWKNZKXNNFCW
|
8.5 | IC50 | 9 | — | |
SJYQOVMGZOATNK
|
8.5 | IC50 | 9 | — | |
SLKHMZQUNIHINK
|
8.5 | IC50 | 10 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
USYASDQVUTWEQM
|
8.5 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
8.5 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
8.5 | IC50 | 9 | — | |
CHADTINFLWZSKR
|
8.5 | Ki | 26 | — | |
JMQCXZBXWOIDIO
|
8.5 | Ki | 9 | — | |
ODNOTLMFNVWFTJ
|
8.5 | Ki | 11 | — | |
SGHXFHRRWFLILP
|
8.5 | Ki | 29 | — |