Target Details
| UniProt AC | Q9H9B1 |
|---|---|
| Gene Symbol | EHMT1 |
| Protein Name | Histone-lysine N-methyltransferase EHMT1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF13637 (Ank_4) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 109
- Clinical molecules 0
- Avg pChEMBL 7.39
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJXNYIVGMQXAMD
|
6.4 | IC50 | 2 | — | |
AHSGGTMURLDJJM
|
6.3 | IC50 | 2 | — | |
LDFAJFPHFKEJOI
|
6.2 | IC50 | 2 | — | |
OSXFATOLZGZLSK
|
6.2 | IC50 | 3 | — | |
DYEFUKCXAQOFHX
|
6.1 | IC50 | 31 | — | |
JBMUWBUCVSKHLE
|
6.1 | Kd | 2 | — | |
YWWZCHLUQSHMCL
|
6.1 | IC50 | 2 | — | |
YRFPHJAMBMALTM
|
6.1 | IC50 | 2 | — | |
TYZFQSLJTWPSDS
|
6.0 | IC50 | 2 | — |