Target Details
| UniProt AC | Q9H9B1 |
|---|---|
| Gene Symbol | EHMT1 |
| Protein Name | Histone-lysine N-methyltransferase EHMT1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF13637 (Ank_4) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 109
- Clinical molecules 0
- Avg pChEMBL 7.39
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTBKCXDRYUDIPI
|
7.5 | IC50 | 2 | — | |
MROKTUUFAWVTEF
|
7.5 | IC50 | 2 | — | |
LNLYAENQQBUQGQ
|
7.5 | IC50 | 2 | — | |
JOHUZOVWSNNWQZ
|
7.5 | IC50 | 2 | — | |
CXHSPDIJBBFXBC
|
7.5 | IC50 | 2 | — | |
PIXKGBJULNYOEX
|
7.5 | IC50 | 2 | — | |
SEIITEYCJLDVFW
|
7.5 | IC50 | 2 | — | |
WGURLEOJEIDTBP
|
7.5 | IC50 | 2 | — | |
XZUWJVJVVBARGQ
|
7.4 | IC50 | 2 | — | |
BKCDJTRMYWSXMC
|
7.4 | IC50 | 3 | — | |
GWCXSYHLYREIAK
|
7.4 | IC50 | 2 | — | |
LSNVRHZIUYXNRN
|
7.4 | IC50 | 2 | — | |
UUFAYOSBAHOCOU
|
7.4 | IC50 | 2 | — | |
GQJJJDCHUVVIMA
|
7.4 | IC50 | 2 | — | |
QAQNPAOMUGDFRD
|
7.4 | IC50 | 2 | — | |
GRCRJEGHKCSKNE
|
7.3 | IC50 | 2 | — | |
FNKMWVAWPMHKHA
|
7.3 | IC50 | 2 | — | |
FGAGTVKUPJXOMV
|
7.3 | IC50 | 2 | — | |
CHEFNBAYIGSOIR
|
7.3 | IC50 | 3 | — | |
OPOCBCGSTOFGIL
|
7.3 | IC50 | 2 | — | |
XIVUGRBSBIXXJE
|
7.3 | IC50 | 2 | — | |
OWORSODZTADOQX
|
7.3 | IC50 | 2 | — | |
NDKARMJRFVQCIS
|
7.3 | IC50 | 2 | — | |
AKOSZLHLQSSJQB
|
7.2 | IC50 | 2 | — | |
NKRNUYLZAXRLJU
|
7.2 | IC50 | 2 | — | |
RBBZOCOZIYNTCM
|
7.2 | IC50 | 2 | — | |
PYGWCVPYKMILCJ
|
7.1 | IC50 | 2 | — | |
ZZSNUOGALFUINV
|
7.1 | IC50 | 2 | — | |
VMVRYCYPSDCNEH
|
7.1 | IC50 | 2 | — | |
FNDUCTFWOZQGTB
|
7.1 | IC50 | 2 | — | |
WGTLTEYVKMNATO
|
7.1 | IC50 | 2 | — | |
FNRUPVONTWZCGL
|
7.1 | IC50 | 2 | — | |
RNAMYOYQYRYFQY
|
7.1 | IC50 | 3 | — | |
YAXJFGYPFUEOCZ
|
7.0 | IC50 | 3 | — | |
DCGOBPRQIYFVOD
|
7.0 | IC50 | 2 | — | |
LMXOHSDXUQEUSF
|
7.0 | IC50 | 6 | — | |
YBKZQRANOVULPZ
|
7.0 | IC50 | 2 | — | |
SFOCRSFKWQNGAT
|
6.9 | IC50 | 2 | — | |
JIPXEHIHQRXFCZ
|
6.8 | IC50 | 2 | — | |
MDFCEIJITSVGGO
|
6.8 | IC50 | 2 | — | |
FQOJFAZVDGPADJ
|
6.7 | IC50 | 3 | — | |
HWEQZXCORSHBDW
|
6.7 | IC50 | 2 | — | |
DRZGMVJAYULHIP
|
6.7 | IC50 | 3 | — | |
ZJUKTBDSGOFHSH
|
6.6 | IC50 | 22 | — | |
GOCBKOQITCNXIM
|
6.6 | IC50 | 2 | — | |
CUXOFABLNDVFGR
|
6.5 | IC50 | 2 | — | |
QHYRXLJGNSPRGA
|
6.5 | IC50 | 2 | — | |
RXNZKWRSWQWERQ
|
6.5 | IC50 | 2 | — | |
XAHHWLRJWBHPFE
|
6.5 | IC50 | 2 | — | |
KKXRBRPMTQSNTJ
|
6.4 | IC50 | 3 | — |