Target Details
| UniProt AC | Q9H9B1 |
|---|---|
| Gene Symbol | EHMT1 |
| Protein Name | Histone-lysine N-methyltransferase EHMT1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF13637 (Ank_4) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 109
- Clinical molecules 0
- Avg pChEMBL 7.39
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VSEYIEDVOXUHFM
|
8.9 | IC50 | 3 | — | |
PZHMEFBKSLGDIS
|
8.8 | IC50 | 3 | — | |
KZOJJUVZAJGNQV
|
8.4 | IC50 | 2 | — | |
GHCDVBSKNGUGCK
|
8.3 | IC50 | 2 | — | |
CZXPVZMKOLPPPQ
|
8.2 | IC50 | 2 | — | |
GKNHULHXRNRLNS
|
8.2 | IC50 | 2 | — | |
SJRUKFZRLQHAEM
|
8.2 | IC50 | 2 | — | |
ZYNUWSFRZCRKSN
|
8.2 | IC50 | 2 | — | |
ONQXWOCNSKDACO
|
8.1 | IC50 | 2 | — | |
YNISGSVZVOGISR
|
8.1 | IC50 | 2 | — | |
FDSPSLJTTWLHQY
|
8.0 | IC50 | 3 | — | |
CHOFEGBVNPOIOH
|
8.0 | IC50 | 2 | — | |
KLWZLAHWDCVBRC
|
8.0 | IC50 | 2 | — | |
QOBAMCAMCSCFMK
|
8.0 | IC50 | 3 | — | |
RZQMLTKBWRSHHE
|
8.0 | IC50 | 3 | — | |
XLDKAPYGJVCXCU
|
8.0 | IC50 | 2 | — | |
ZDINBSHEURZXDD
|
8.0 | IC50 | 2 | — | |
AEJULKFUIXWPOX
|
7.9 | IC50 | 2 | — | |
AFFYALXSRBVAPQ
|
7.9 | IC50 | 2 | — | |
AUFSXIYCIRDGIZ
|
7.9 | IC50 | 2 | — | |
MLTCNEHPZTWJKH
|
7.9 | IC50 | 2 | — | |
PGVIWADEDHEJGB
|
7.9 | IC50 | 2 | — | |
UQBQMWLGFSNAIR
|
7.8 | IC50 | 2 | — | |
VWFQZXWQZKXLEI
|
7.8 | IC50 | 2 | — | |
LNFNHVCQOOPPAK
|
7.8 | IC50 | 2 | — | |
VAAQORJZPYRYHH
|
7.8 | IC50 | 2 | — | |
NDEREOOBAVLGBN
|
7.8 | IC50 | 2 | — | |
RCWUUMJJJVFQSV
|
7.8 | IC50 | 2 | — | |
GLDHWRNHMTWDKJ
|
7.7 | IC50 | 2 | — | |
NEHZFWWDTWSDKX
|
7.7 | IC50 | 2 | — | |
RINVPEJSDRLKKC
|
7.7 | IC50 | 2 | — | |
AULLUGALUBVBDD
|
7.7 | IC50 | 2 | — | |
AVSMKKGLVDCOEU
|
7.7 | IC50 | 2 | — | |
KGUAKPWBXICIMX
|
7.7 | IC50 | 2 | — | |
NYDFIFBPOWTDSS
|
7.7 | IC50 | 2 | — | |
QOECJCJVIMVJGX
|
7.7 | IC50 | 8 | — | |
YBQHFHPOKHPBRB
|
7.7 | IC50 | 2 | — | |
DJKVIUVJRXEKNV
|
7.7 | IC50 | 2 | — | |
GDWIBPWOSOTLGZ
|
7.7 | IC50 | 2 | — | |
WLSUJPBXUGENOU
|
7.7 | IC50 | 2 | — | |
OIHAWFCPBDLPLR
|
7.7 | IC50 | 3 | — | |
MEVMMQQJOXBSAX
|
7.6 | IC50 | 2 | — | |
YMSMSNAIHUSOEZ
|
7.6 | IC50 | 2 | — | |
YQVURWXJUBXXCZ
|
7.6 | IC50 | 2 | — | |
FKTQPAVLUZRKHC
|
7.6 | IC50 | 2 | — | |
LHNQVGYVOOWUCA
|
7.6 | IC50 | 2 | — | |
AUGGZTSGLVEWLK
|
7.6 | IC50 | 2 | — | |
MFOQRJHECLPWDG
|
7.6 | IC50 | 2 | — | |
PZFSXMLFZTZWAI
|
7.6 | IC50 | 2 | — | |
YTZXLVDHUCDBOG
|
7.6 | IC50 | 2 | — |