Target Details
| UniProt AC | Q9H8M2 |
|---|---|
| Gene Symbol | BRD9 |
| Protein Name | Bromodomain-containing protein 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF12024 (DUF3512) |
Summary
- Multi-target molecules 111
- Clinical molecules 0
- Avg pChEMBL 7.15
KEGG Pathways (1)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OJEWEVFWZJYOCQ
|
7.3 | IC50 | 2 | — | |
OPPFAMQHKKPXOS
|
7.3 | IC50 | 2 | — | |
OTCCCUQXFNXOEA
|
7.3 | IC50 | 2 | — | |
PMLQWYVXIXUHRE
|
7.3 | IC50 | 2 | — | |
PXCPUAMIKTYRQJ
|
7.3 | IC50 | 2 | — | |
RNLLYKSZEHIACO
|
7.3 | IC50 | 2 | — | |
SGIKXXJDVXGQMZ
|
7.3 | IC50 | 2 | — | |
SZYWJNANYDZYKI
|
7.3 | IC50 | 2 | — | |
TYYUGGGBAYVOOY
|
7.3 | IC50 | 2 | — | |
UTWBAQAOZKWZEZ
|
7.3 | IC50 | 2 | — | |
VALZAYGWSVKVKA
|
7.3 | IC50 | 2 | — | |
VUQFCAKQINYQAI
|
7.3 | IC50 | 2 | — | |
VXPZXQXSSMBLQQ
|
7.3 | IC50 | 2 | — | |
WSSCIZFVUUISJR
|
7.3 | IC50 | 2 | — | |
XAYVOLACEOYNKF
|
7.3 | IC50 | 2 | — | |
XQSOXJOPLWACDH
|
7.3 | IC50 | 2 | — | |
GQTWFQWDINXZPP
|
7.2 | IC50 | 2 | — | |
UXFKGTAATGRBOW
|
7.2 | Ki | 2 | — | |
KPWWFNXRLAAREN
|
7.2 | Kd | 12 | — | |
AFNYOROEWXANDC
|
7.2 | Kd | 2 | — | |
DDHSJBNVVYBOFE
|
7.2 | Kd | 2 | — | |
DGJREYHVQYZTEV
|
7.2 | Kd | 6 | — | |
AIOCFZJGGGEWDK
|
7.1 | IC50 | 2 | — | |
HONYBLSJNSYWKQ
|
7.0 | IC50 | 3 | — | |
LVDRREOUMKACNJ
|
7.0 | Kd | 2 | — | |
LBUBPCSKFDKKFO
|
6.9 | IC50 | 2 | — | |
NMMSMXOCHXLFTJ
|
6.9 | IC50 | 2 | — | |
WCRAZRPWWUJMQW
|
6.9 | Ki | 2 | — | |
DLOWILGTRNUHPQ
|
6.8 | Kd | 2 | — | |
RJEMCUZKQLRUIS
|
6.8 | IC50 | 4 | — | |
UYBRROMMFMPJAN
|
6.8 | IC50 | 8 | — | |
LQDXWIYREJVTTB
|
6.8 | IC50 | 4 | — | |
WLUMGCPGWDQOSB
|
6.7 | IC50 | 3 | — | |
MREZOHBMPINXNX
|
6.7 | IC50 | 2 | — | |
RORQWFZBNDBULQ
|
6.6 | Kd | 3 | — | |
YHMNROQTPUKNLA
|
6.6 | IC50 | 8 | — | |
SPSRAFOXVSNAJA
|
6.5 | IC50 | 3 | — | |
GACUWBJOGWUMHF
|
6.5 | Kd | 2 | — | |
BMVCSXFOQPYKKC
|
6.5 | IC50 | 5 | — | |
MYFFGZYMLKZBPZ
|
6.5 | IC50 | 4 | — | |
ZJBYPBSYPDAGHO
|
6.5 | Ki | 2 | — | |
COGXRBWRVXDPDM
|
6.4 | IC50 | 2 | — | |
ZACGKNYCBHUCNI
|
6.3 | IC50 | 2 | — | |
DDRHNLQKGDBMGK
|
6.3 | Kd | 2 | — | |
YJIKHWNQMIOYBT
|
6.3 | IC50 | 2 | — | |
AZCFROYDWGJIHI
|
6.2 | IC50 | 3 | — | |
APJDTDALQSVARU
|
6.2 | IC50 | 3 | — | |
BFTKDWYIRJGJCA
|
6.1 | IC50 | 3 | — | |
CBGFEMSXMIJQKG
|
6.1 | IC50 | 3 | — | |
NRTSFXVZIHRSAM
|
6.1 | IC50 | 2 | — |