Target Details
| UniProt AC | Q9H8M2 |
|---|---|
| Gene Symbol | BRD9 |
| Protein Name | Bromodomain-containing protein 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF12024 (DUF3512) |
Summary
- Multi-target molecules 111
- Clinical molecules 0
- Avg pChEMBL 7.15
KEGG Pathways (1)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIUXKWFQVPTMEQ
|
9.6 | Kd | 3 | — | |
UOQAFGWMKNIVAR
|
9.3 | Kd | 6 | — | |
PMWIFIWWNULSSP
|
8.7 | Kd | 2 | — | |
AVBQIZYXLUVYRI
|
8.5 | IC50 | 2 | — | |
FWTDDBIMDSVPTR
|
8.4 | IC50 | 2 | — | |
FQZLYYSRDPJOHB
|
8.4 | Kd | 2 | — | |
IHZXYEFDJOXHGJ
|
8.3 | IC50 | 2 | — | |
BQAKOVGAYWUDIT
|
8.2 | IC50 | 3 | — | |
QVMOJFHRHLLSOT
|
8.2 | IC50 | 3 | — | |
KCZMLIMZGLNMQN
|
8.1 | IC50 | 2 | — | |
MOYOGONDTNZILF
|
8.0 | IC50 | 2 | — | |
WHKOQEHRVJBOCH
|
8.0 | IC50 | 2 | — | |
ZAGCLFXBHOXXEN
|
7.9 | Kd | 4 | — | |
TWAMSFSFBGEKAM
|
7.9 | IC50 | 2 | — | |
ZJDRXPZROJHILR
|
7.9 | IC50 | 2 | — | |
POICMTYCJMMADL
|
7.9 | IC50 | 3 | — | |
BJFSUDWKXGMUKA
|
7.8 | Kd | 3 | — | |
RBUYFHLQNPJMQM
|
7.8 | Kd | 10 | — | |
RPMQBLMPGMFXLD
|
7.8 | Kd | 4 | — | |
JGOZUFGBTSAWEI
|
7.6 | IC50 | 4 | — | |
UIULTDHSORWSLL
|
7.5 | IC50 | 2 | — | |
RPBMXJHQYJLPDN
|
7.5 | Kd | 2 | — | |
AAAQFGUYHFJNHI
|
7.5 | IC50 | 252 | — | |
GVJYOLRRZZUUOE
|
7.5 | IC50 | 5 | — | |
JSTVWXBDEJQXEC
|
7.4 | IC50 | 2 | — | |
SZKYAPUMPFTJEP
|
7.4 | IC50 | 2 | — | |
WRUWGLUCNBMGPS
|
7.4 | IC50 | 5 | — | |
YTQRBAXLTKDECT
|
7.4 | Ki | 5 | — | |
OAXPZAPALNMAIG
|
7.3 | IC50 | 2 | — | |
AGAONEPKOIFRDY
|
7.3 | IC50 | 2 | — | |
ALGGNHJBKHNFCV
|
7.3 | IC50 | 2 | — | |
BGFQTYLHACMCNL
|
7.3 | IC50 | 2 | — | |
BMSMDNAPNHYSPD
|
7.3 | IC50 | 2 | — | |
BXQXTJBUXHEDIJ
|
7.3 | IC50 | 2 | — | |
BXZKFTOWUAMBMJ
|
7.3 | IC50 | 2 | — | |
CCJMJJQREOHGIP
|
7.3 | IC50 | 2 | — | |
DDGMMVZOQQXROR
|
7.3 | IC50 | 2 | — | |
DPQPWJKNLZNKIJ
|
7.3 | IC50 | 2 | — | |
DUZIGRKTZUROMM
|
7.3 | IC50 | 2 | — | |
FQLVQDGNXPTTNU
|
7.3 | IC50 | 2 | — | |
HFAUIBUNFUHOCA
|
7.3 | IC50 | 2 | — | |
IKEOGNMNDJHWOI
|
7.3 | IC50 | 2 | — | |
JESNLPWFJFGFAG
|
7.3 | IC50 | 2 | — | |
KGAFBKKTQDWRLO
|
7.3 | IC50 | 2 | — | |
KVFUIRXLUZSQDJ
|
7.3 | IC50 | 2 | — | |
KWTLWVFVCIQSGS
|
7.3 | IC50 | 2 | — | |
LOPDQTRAACJHKL
|
7.3 | IC50 | 2 | — | |
MOXDTUJERWXKNZ
|
7.3 | IC50 | 2 | — | |
NCHWRSJTCVNFGY
|
7.3 | IC50 | 2 | — | |
NEVWSLOXJDXDEC
|
7.3 | IC50 | 2 | — |