Target Details
| UniProt AC | Q9H4B4 |
|---|---|
| Gene Symbol | PLK3 |
| Protein Name | Serine/threonine-protein kinase PLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 203
- Clinical molecules 24
- Avg pChEMBL 6.88
KEGG Pathways (3)
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AGYRJOAGMDIFKL
|
6.2 | Ki | 17 | — | |
DZIPQNPWTUXXSJ
|
6.2 | Ki | 18 | — | |
GILNGUYOGYOZMP
|
6.2 | IC50 | 6 | — | |
KWSZYBNXNYRQCC
|
6.2 | Ki | 21 | — | |
NWAUBAGBGOPJLF
|
6.2 | Ki | 51 | Yes | |
RWEHAHIEUDLKGT
|
6.2 | Ki | 33 | — | |
UGEJLCNSVIVALC
|
6.2 | Ki | 41 | — | |
UUWNXFJBBYAMDT
|
6.2 | Ki | 46 | — | |
XIOOJUQFJYPVLA
|
6.2 | Ki | 17 | — | |
YRUKXDLUMKDTLG
|
6.2 | IC50 | 2 | — | |
LDFXILCAFQHTNH
|
6.2 | IC50 | 3 | — | |
HFNKQEVNSGCOJV
|
6.2 | Kd | 65 | — | |
KMZDOKNRRSNTSW
|
6.2 | IC50 | 2 | — | |
UZVJWQPORUUHRW
|
6.1 | IC50 | 3 | — | |
ZHJGWYRLJUCMRT
|
6.1 | Kd | 18 | — | |
MLSKNMPNUOPUAB
|
6.1 | IC50 | 3 | — | |
FTFDOZLQPLTYBX
|
6.1 | IC50 | 7 | Yes | |
AWJPVXSHMIELNJ
|
6.1 | Ki | 23 | — | |
BQPLWJRDSDNGNE
|
6.1 | Ki | 16 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
GFOMFROIIBQABZ
|
6.1 | Ki | 7 | — | |
GQHSVFWCNBWKGM
|
6.1 | Ki | 3 | — | |
GWJHMRBQEUHFOC
|
6.1 | Ki | 42 | — | |
HSKVRPZJBMXFDX
|
6.1 | Ki | 20 | — | |
IOBVCHJTLVPPBR
|
6.1 | Ki | 39 | — | |
OKCNACDPDSQZSE
|
6.1 | Ki | 7 | — | |
OLVBAUVSICCWEJ
|
6.1 | Ki | 39 | — | |
UPITUWGOTMBQLX
|
6.1 | Ki | 13 | — | |
YQKSNDNARJQAHP
|
6.1 | Ki | 12 | — | |
ZQVQTUFEKLITNT
|
6.1 | Ki | 10 | — | |
HKSZLNNOFSGOKW
|
6.0 | Kd | 213 | — | |
WQQABBZFVHSXMU
|
6.0 | IC50 | 3 | — | |
BSFNGHCTZDCQBF
|
6.0 | Ki | 3 | — | |
KSMYGTHXVJXRTI
|
6.0 | IC50 | 3 | — | |
AJJBWPRLFOMJCY
|
6.0 | IC50 | 3 | — | |
CXPHUBRUHJPONW
|
6.0 | IC50 | 3 | — | |
IJDPNONZYDDAHT
|
6.0 | IC50 | 3 | — | |
AYJBHLUSGLQYDG
|
6.0 | Ki | 16 | — | |
AZTMYWWWILJAKW
|
6.0 | Ki | 16 | Yes | |
CSMDANWISUYBHA
|
6.0 | Ki | 8 | — | |
HATNHAMXMKJCEI
|
6.0 | Ki | 9 | — | |
IQNOGQGSOHNMCL
|
6.0 | Ki | 14 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KBRJIBFRLFVYJL
|
6.0 | Ki | 5 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LRLDYTTWQIFWBD
|
6.0 | Ki | 25 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NEWAULHLLUCDPD
|
6.0 | Ki | 27 | — | |
RJZDECGDCKOHBV
|
6.0 | Ki | 70 | — | |
SPMHGQZFMNZCBV
|
6.0 | Ki | 30 | Yes |