Target Details
| UniProt AC | Q9H4B4 |
|---|---|
| Gene Symbol | PLK3 |
| Protein Name | Serine/threonine-protein kinase PLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 203
- Clinical molecules 24
- Avg pChEMBL 6.88
KEGG Pathways (3)
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNCCSJOQZGLCIQ
|
6.8 | IC50 | 3 | — | |
GSXMJWLLQORXFR
|
6.8 | IC50 | 3 | — | |
NERSFQYNEXMEPK
|
6.8 | IC50 | 3 | — | |
JPWPZFYYVIFSAZ
|
6.8 | IC50 | 3 | — | |
QMGCOLHGTKYVOP
|
6.7 | IC50 | 3 | — | |
KTQYQHLIMZOBSM
|
6.7 | Ki | 12 | — | |
SFNMDOXBLCGZMQ
|
6.7 | IC50 | 3 | — | |
YXRJOXHIGGNCBU
|
6.7 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
6.7 | IC50 | 408 | — | |
HLHNFPFYQRRGPP
|
6.6 | IC50 | 2 | — | |
XEXSGNRGTBSSOU
|
6.6 | IC50 | 3 | — | |
BNLPAUPVSCPTDM
|
6.6 | Ki | 15 | — | |
GWMATETWMAQOFL
|
6.6 | Ki | 36 | — | |
HLHNFPFYQRRGPP
|
6.6 | IC50 | 2 | — | |
NLUPJKQOKWBWFC
|
6.6 | Ki | 69 | — | |
OWRXHGAFWZFFCW
|
6.6 | Ki | 113 | — | |
DZSUJUOJJJCWGG
|
6.6 | Ki | 55 | Yes | |
INCAIRNHZBEWOA
|
6.6 | IC50 | 5 | Yes | |
SWIVJTVGOIXUKC
|
6.6 | IC50 | 9 | — | |
ZDQJNYLFGPXANH
|
6.5 | IC50 | 3 | — | |
MCCCQFAOMZMZKE
|
6.5 | Ki | 52 | — | |
DFKJNGVBNCASDM
|
6.5 | IC50 | 2 | — | |
UXNCNPVLRQGOMH
|
6.5 | IC50 | 3 | — | |
SLGRRBVHGIPHNQ
|
6.5 | IC50 | 2 | — | |
NCCZKHZUPCPIOT
|
6.4 | IC50 | 3 | — | |
NTVFVNYEAMJGDF
|
6.4 | IC50 | 3 | — | |
GUMBHNMWKMFKRT
|
6.4 | Ki | 23 | — | |
PJUVRETYCLPAFV
|
6.4 | Ki | 20 | — | |
PUPCRRRSBUYJAD
|
6.4 | Ki | 44 | Yes | |
VNGYQBMDQMDALH
|
6.4 | Ki | 25 | — | |
AILANCLYZDKELS
|
6.4 | IC50 | 3 | — | |
OSCRFGZIFNWYIZ
|
6.4 | IC50 | 3 | — | |
RJERVODZSCACGJ
|
6.4 | IC50 | 3 | — | |
JKZKKHVTLCFCGS
|
6.3 | IC50 | 3 | — | |
MOSNATYSIYEVTF
|
6.3 | IC50 | 2 | — | |
MRITYVDXXFOOAU
|
6.3 | Kd | 6 | — | |
KSNXWDGHPBZSBU
|
6.3 | IC50 | 2 | — | |
QIMUQYHRHHNTNY
|
6.3 | IC50 | 3 | — | |
BSFNGHCTZDCQBF
|
6.3 | Ki | 93 | — | |
DKXHSOUZPMHNIZ
|
6.3 | Ki | 51 | Yes | |
MVJMMLFMPWITEJ
|
6.3 | Ki | 110 | — | |
PYXQMJSGJIJHJT
|
6.3 | Ki | 28 | — | |
ZCCJKVBTHCOISJ
|
6.3 | Ki | 46 | — | |
OPJOIUDMJCRLNO
|
6.3 | IC50 | 2 | — | |
ZAJAQZFUONWQPQ
|
6.3 | IC50 | 3 | — | |
BRLRIFFHVZNKFH
|
6.2 | IC50 | 2 | — | |
GHPFSYCYZJKVDZ
|
6.2 | Ki | 18 | Yes | |
VVQWZQWJWMTPJY
|
6.2 | IC50 | 2 | — | |
VVQWZQWJWMTPJY
|
6.2 | IC50 | 2 | — |