Target Details
| UniProt AC | Q9H4B4 |
|---|---|
| Gene Symbol | PLK3 |
| Protein Name | Serine/threonine-protein kinase PLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 203
- Clinical molecules 24
- Avg pChEMBL 6.88
KEGG Pathways (3)
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DKSNLQYRZJKYOC
|
7.4 | Ki | 51 | — | |
YIJGUCDNKKHCPF
|
7.4 | IC50 | 2 | — | |
CVLJBLIMHPEZJC
|
7.4 | IC50 | 2 | — | |
FTVMYIRRFFYFIH
|
7.4 | IC50 | 3 | — | |
UHCHLTQBLNUYRT
|
7.4 | IC50 | 2 | — | |
VZDOSGQBGHVVCU
|
7.3 | IC50 | 3 | — | |
VINNOSMQDSWDTC
|
7.3 | IC50 | 3 | — | |
QDLHCMPXEPAAMD
|
7.3 | IC50 | 13 | Yes | |
LYNBNVBMAGDJRW
|
7.3 | Ki | 81 | — | |
TVENGSGQLJMALI
|
7.3 | Ki | 2 | — | |
ZRGJZUSQJGUWJC
|
7.3 | IC50 | 2 | — | |
GYDZFEKAOMUPJL
|
7.3 | IC50 | 2 | — | |
SXNJFOWDRLKDSF
|
7.2 | IC50 | 3 | — | |
SXNJFOWDRLKDSF
|
7.2 | IC50 | 8 | — | |
JVAPIYLPNKDKAQ
|
7.2 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
7.2 | Ki | 63 | — | |
SRUYMJRFVGLQDV
|
7.2 | Ki | 37 | — | |
ZXLFIHLBHMLHFJ
|
7.2 | Ki | 31 | — | |
MYVQSDVXBZNNLF
|
7.2 | IC50 | 8 | Yes | |
JETXRGKNZYUPEF
|
7.2 | IC50 | 6 | — | |
GGHUWFIXZDQNHR
|
7.1 | IC50 | 8 | Yes | |
GDMBPOYBSJXINX
|
7.1 | IC50 | 2 | — | |
JCFJQIHDZHHMQT
|
7.1 | Ki | 42 | — | |
KKYPRNBBPBRJQX
|
7.1 | Ki | 40 | — | |
KPDOBADQSPMGFP
|
7.1 | IC50 | 3 | — | |
UEIRKXUBXCSHJE
|
7.1 | Ki | 19 | — | |
ZBJWJVGFIIULBV
|
7.1 | IC50 | 3 | — | |
MVYFNZROIDKPOZ
|
7.1 | IC50 | 3 | — | |
HOOQLZPFGONGJY
|
7.0 | IC50 | 3 | — | |
MAULBJVKJOGNGD
|
7.0 | IC50 | 3 | — | |
URBLFMVEDFWKGZ
|
7.0 | IC50 | 6 | — | |
LKUJDAHYLPICSE
|
7.0 | Ki | 24 | — | |
OWDRQHVEJIYVOI
|
7.0 | Ki | 47 | — | |
QKPLUKMJEKRAJD
|
7.0 | Ki | 30 | Yes | |
NUQUWKXNHFMEAJ
|
7.0 | IC50 | 3 | — | |
CAVRDKDHKZOOIF
|
7.0 | IC50 | 3 | — | |
AAWUJXDNCDOXTN
|
6.9 | IC50 | 3 | — | |
WPPGBVWZGMDXKF
|
6.9 | IC50 | 5 | — | |
HWIAWKKIXLIVDB
|
6.9 | IC50 | 2 | — | |
ITAJXWHXKVYGCF
|
6.9 | Ki | 5 | — | |
PVVRSMIEEGPASF
|
6.9 | IC50 | 3 | — | |
JQRWYCWILFBHJT
|
6.8 | IC50 | 7 | Yes | |
ANAAVHLLZPPWCU
|
6.8 | IC50 | 6 | — | |
ITYGFIRONBGARW
|
6.8 | IC50 | 3 | — | |
UEILKDPTXUZCFH
|
6.8 | IC50 | 3 | — | |
FVLMDPWEHBGZDD
|
6.8 | IC50 | 3 | — | |
NCDFJOWBEBTLBV
|
6.8 | IC50 | 2 | — | |
MJLKHAZEWYICMC
|
6.8 | Ki | 4 | — | |
PGHXJQMSVOKZRE
|
6.8 | IC50 | 3 | — | |
RKWOVOVDWBRGQO
|
6.8 | Kd | 5 | — |