Target Details
| UniProt AC | Q9H3Y6 |
|---|---|
| Gene Symbol | SRMS |
| Protein Name | Tyrosine-protein kinase Srms |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 71
- Clinical molecules 7
- Avg pChEMBL 6.81
Active Molecules (71)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CFIBXVQLBVNOHW
|
6.2 | Ki | 64 | — | |
MIKAKZKNMYZLDX
|
6.2 | Ki | 42 | — | |
NFMGZVPRGVERNN
|
6.2 | Ki | 44 | — | |
STISJUSFFZAZMP
|
6.2 | Ki | 7 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 213 | — | |
BNLPAUPVSCPTDM
|
6.1 | Ki | 15 | — | |
FUMCKNCUEAQHCV
|
6.1 | Ki | 103 | — | |
JXNMCDLXYWQTIW
|
6.1 | Ki | 13 | — | |
UYJNQQDJUOUFQJ
|
6.1 | Ki | 68 | — | |
XKZQZMSAWVDRSP
|
6.1 | Ki | 39 | Yes | |
UIARLYUEJFELEN
|
6.1 | Kd | 289 | Yes | |
AIQDZMUPVYDVLB
|
6.0 | Ki | 48 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KJVWCDAPVMWKLJ
|
6.0 | Ki | 20 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OWFXKTOLFUQPDJ
|
6.0 | Ki | 36 | — | |
WFTZMAAMCVPJJT
|
6.0 | Ki | 26 | — | |
XFWUTMHVDGPWLH
|
6.0 | Ki | 75 | — | |
ZVWRFVCNQOECJS
|
6.0 | Ki | 71 | — |