Target Details
| UniProt AC | Q9H3Y6 |
|---|---|
| Gene Symbol | SRMS |
| Protein Name | Tyrosine-protein kinase Srms |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 71
- Clinical molecules 7
- Avg pChEMBL 6.81
Active Molecules (71)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FDVSOQRNTAPCHB
|
8.2 | Ki | 40 | — | |
FUZSHLVNKZZEKR
|
8.1 | IC50 | 16 | — | |
SRSQULBCTWSVKL
|
8.0 | IC50 | 15 | — | |
ZBNZXTGUTAYRHI
|
7.9 | Kd | 102 | Yes | |
CDISOBGWDHAHGF
|
7.8 | IC50 | 16 | — | |
OMIQRSKHABIPRH
|
7.8 | IC50 | 15 | — | |
CXQHYVUVSFXTMY
|
7.8 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.7 | Kd | 149 | — | |
OPHSZSZDICRBPP
|
7.7 | IC50 | 16 | — | |
YZDJQTHVDDOVHR
|
7.7 | Kd | 23 | — | |
JUSWPUDQOKINJO
|
7.6 | IC50 | 16 | — | |
XYFZVVYVIFJBIS
|
7.6 | IC50 | 17 | — | |
SRUYMJRFVGLQDV
|
7.6 | Ki | 37 | — | |
WPHKIQPVPYJNAX
|
7.6 | Ki | 81 | — | |
XJSFDMGICAWQFS
|
7.6 | Ki | 60 | — | |
AHBFBRPGNOVEBK
|
7.5 | IC50 | 11 | — | |
LSJWYMSFUWBGPN
|
7.3 | IC50 | 17 | — | |
XKFTZKGMDDZMJI
|
7.3 | Ki | 56 | — | |
XOOAAYRIVATZNM
|
7.3 | Ki | 55 | — | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
WMMNTQFZCHUZSM
|
7.2 | IC50 | 14 | — | |
GZYUJXFTHLKPAK
|
7.2 | IC50 | 16 | — | |
NZJCXRPMZJGVCC
|
7.2 | Kd | 8 | — | |
ODPGGGTTYSGTGO
|
7.1 | Kd | 153 | — | |
LAUHLGUSVSJYCI
|
7.1 | IC50 | 16 | — | |
ZGDSBEUMPIMXBM
|
7.1 | Ki | 42 | — | |
VTJHGMZHVOXJPG
|
7.1 | IC50 | 15 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
WDTHDWKPTWWHLS
|
7.0 | IC50 | 13 | — | |
CEUSZLVORFRBCV
|
6.9 | IC50 | 13 | — | |
GXJSLIOOPZRPEV
|
6.9 | Ki | 34 | — | |
UUWNXFJBBYAMDT
|
6.9 | Ki | 46 | — | |
CXBBWVXSZINRCS
|
6.8 | Ki | 41 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
ZWVZORIKUNOTCS
|
6.8 | Ki | 69 | — | |
BIKYDWLMTPRSQL
|
6.7 | Ki | 50 | — | |
XNEPVLVYFUGJLF
|
6.7 | Ki | 27 | — | |
MVJMMLFMPWITEJ
|
6.6 | Ki | 110 | — | |
XHORJSJFHVABEA
|
6.6 | Ki | 49 | — | |
VKBFHTIUXUCYRQ
|
6.5 | Ki | 66 | — | |
XBYVOPRDASFDMY
|
6.5 | Ki | 42 | — | |
WVXNSAVVKYZVOE
|
6.4 | IC50 | 92 | — | |
HCNIBOQWDVOZKF
|
6.4 | Ki | 26 | — | |
PQNWNVWJXPSZFR
|
6.4 | Ki | 21 | — | |
SHPFDGWALWEPGS
|
6.4 | Kd | 35 | — | |
JSDGKSMNPHJDFK
|
6.3 | Ki | 35 | — | |
ZVPDNRVYHLRXLX
|
6.3 | Ki | 35 | Yes | |
VAARYSWULJUGST
|
6.2 | Kd | 119 | Yes | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — |