Target Details
| UniProt AC | Q9H300 |
|---|---|
| Gene Symbol | PARL |
| Protein Name | Presenilin-associated rhomboid-like protein, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01694 (Rhomboid) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 7.46
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
8.3 | Kd | 599 | — | |
YFGBSZIJBXPJHD
|
7.5 | IC50 | 2 | — | |
WSGJLZWGFILROL
|
7.4 | IC50 | 2 | — | |
JGLCCKSTFKAEJE
|
7.3 | IC50 | 2 | — | |
LXWDSHFLPIJHPM
|
7.3 | IC50 | 2 | — | |
QPVPBCXDMKGAQP
|
7.2 | IC50 | 2 | — | |
GRZBUTPJWIBTNF
|
7.2 | IC50 | 2 | — |