Target Details
| UniProt AC | Q9H2X6 |
|---|---|
| Gene Symbol | HIPK2 |
| Protein Name | Homeodomain-interacting protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 256
- Clinical molecules 15
- Avg pChEMBL 6.86
KEGG Pathways (1)
Active Molecules (256)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HMKKDSBJGMESJD
|
6.3 | Ki | 10 | — | |
IABDKYMGRMDGMM
|
6.3 | Ki | 10 | — | |
JWQOJVOKBAAAAR
|
6.3 | Ki | 29 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
QQXBOOIPHBWOGC
|
6.3 | Ki | 4 | — | |
RYYNGWLOYLRZLK
|
6.3 | Ki | 104 | — | |
YGUMGYOBTNGZKS
|
6.3 | Ki | 12 | — | |
YKJSWMAVAKRUAN
|
6.3 | Ki | 19 | — | |
LHNIIDJUOCFXAP
|
6.3 | Kd | 20 | Yes | |
OSVUGUHRKMMBSE
|
6.2 | Kd | 170 | — | |
HZGYSSZTTMUCJE
|
6.2 | Ki | 8 | — | |
KAICHBSRWFIESE
|
6.2 | Ki | 14 | — | |
LRZYYIZFBXFSJB
|
6.2 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
6.2 | Ki | 41 | — | |
OWDRQHVEJIYVOI
|
6.2 | Ki | 47 | — | |
PMXPVPGZZRMXIV
|
6.2 | Ki | 8 | — | |
SRONQUHCRFZABC
|
6.2 | Ki | 28 | — | |
SYLTYCLPHHSEIJ
|
6.2 | Ki | 27 | — | |
XYZNKCSDQRKAFR
|
6.2 | Ki | 53 | — | |
PXEZKQRPUIYVRE
|
6.2 | IC50 | 2 | — | |
AXRCEOKUDYDWLF
|
6.1 | Kd | 31 | — | |
GQLWKGVBOIYMTN
|
6.1 | Ki | 35 | — | |
GSXRCPJTNIGKSZ
|
6.1 | Ki | 43 | — | |
JZTOUVBEZONDKA
|
6.1 | Ki | 80 | — | |
MCCCQFAOMZMZKE
|
6.1 | Ki | 52 | — | |
PDBPUXLUVDSLML
|
6.1 | Ki | 14 | — | |
TZSJMSZEKQGCBI
|
6.1 | Ki | 15 | — | |
WYCBJBMCGVVCMY
|
6.1 | Ki | 8 | — | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
YEKVTSRZMPLPFK
|
6.1 | Ki | 17 | — | |
YOVNFNXUCOWYSG
|
6.1 | Ki | 33 | Yes | |
YRVHWCZERXVDLL
|
6.1 | Ki | 6 | — | |
ASZYLQGAFPWILY
|
6.0 | IC50 | 2 | — | |
CYLYPHIGBMPKCK
|
6.0 | Ki | 6 | — | |
GNRAZHYXXNIXFM
|
6.0 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.0 | Kd | 65 | — | |
HOBMVEVXDIOMDM
|
6.0 | Ki | 18 | — | |
IOYGZJJCJBOPDM
|
6.0 | Ki | 8 | — | |
IUEBPIPDFMCSTP
|
6.0 | Ki | 29 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JIYNLLZDWHPTOM
|
6.0 | Ki | 5 | — | |
JOOXLOJCABQBSG
|
6.0 | Kd | 139 | — | |
KDYPNLAUCVXSFG
|
6.0 | IC50 | 2 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MTCHQDWUHQADSY
|
6.0 | Ki | 29 | — | |
NRGYZNJPCGRCLV
|
6.0 | Ki | 52 | — | |
OADRBDVURCEKRP
|
6.0 | Ki | 44 | — | |
QNUKRWAIZMBVCU
|
6.0 | Ki | 46 | — | |
SFJKSVOPZBRMLV
|
6.0 | IC50 | 2 | — |