Target Details
| UniProt AC | Q9H2X6 |
|---|---|
| Gene Symbol | HIPK2 |
| Protein Name | Homeodomain-interacting protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 256
- Clinical molecules 15
- Avg pChEMBL 6.86
KEGG Pathways (1)
Active Molecules (256)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWAUBAGBGOPJLF
|
6.7 | Ki | 51 | Yes | |
XBDWKVLCDCUNHH
|
6.7 | Ki | 18 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
YJBNTRQKJQHMTM
|
6.7 | Ki | 11 | — | |
BPNUQXPIQBZCMR
|
6.7 | Kd | 83 | Yes | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
BPNUQXPIQBZCMR
|
6.6 | Ki | 60 | — | |
CALAEFSQWBJMDU
|
6.6 | Ki | 21 | — | |
CNTCGRJDUJEUDG
|
6.6 | Ki | 37 | — | |
DBKQWGCVGCVPIP
|
6.6 | Ki | 21 | — | |
KYACBMRLQMEIAI
|
6.6 | Ki | 30 | — | |
LXVBELDBJGYFEM
|
6.6 | Ki | 20 | — | |
MNEBTNXXCJJUOW
|
6.6 | Ki | 7 | — | |
ORRHVRJUSPCILV
|
6.6 | Ki | 16 | — | |
RJZDECGDCKOHBV
|
6.6 | Ki | 70 | — | |
WINHZLLDWRZWRT
|
6.6 | Ki | 66 | — | |
ZGDSBEUMPIMXBM
|
6.6 | Ki | 42 | — | |
BWUOLNXJAQPJKF
|
6.6 | IC50 | 7 | — | |
TUVCWJQQGGETHL
|
6.5 | Kd | 22 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
ACNCCUVYXQGPKZ
|
6.5 | Ki | 31 | — | |
BHSOPYVVEZFHDB
|
6.5 | Ki | 25 | Yes | |
CHQYAWLKOUOTQO
|
6.5 | IC50 | 20 | — | |
ISVHLTLEHRZKJC
|
6.5 | Ki | 19 | — | |
OWRXHGAFWZFFCW
|
6.5 | Ki | 113 | — | |
UDRXOUVRNMKWQA
|
6.5 | Ki | 8 | — | |
ULHGAQSVFPOUDY
|
6.5 | Ki | 43 | — | |
UOOZSMNSBYVUGZ
|
6.5 | Ki | 32 | — | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
VNGYQBMDQMDALH
|
6.5 | Ki | 25 | — | |
ZXLFIHLBHMLHFJ
|
6.5 | Ki | 31 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
ODCXYSYHXJMMPY
|
6.5 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
6.4 | Kd | 289 | Yes | |
KGPGFQWBCSZGEL
|
6.4 | Kd | 59 | Yes | |
DYSRECIVMDGUQU
|
6.4 | Ki | 29 | — | |
GUMBHNMWKMFKRT
|
6.4 | Ki | 23 | — | |
JCFJQIHDZHHMQT
|
6.4 | Ki | 42 | — | |
JMQCXZBXWOIDIO
|
6.4 | Ki | 9 | — | |
OQHALFBQFMAXFZ
|
6.4 | Ki | 9 | — | |
PTVPBWWDGZSEAF
|
6.4 | Ki | 63 | — | |
PWIKZIKRKUUHRB
|
6.4 | Ki | 9 | — | |
QONPPIZSNSSCSK
|
6.4 | Ki | 45 | Yes | |
RGOPHVZLEMGMBZ
|
6.4 | Ki | 20 | — | |
XCHWBXBDZRJVDP
|
6.4 | Ki | 51 | — | |
XKZINYYXWJEYEL
|
6.4 | Ki | 37 | — | |
OHHWUWXPWKJQHC
|
6.4 | IC50 | 2 | — | |
JOZUGIHTSIWTIK
|
6.3 | IC50 | 4 | — | |
CIUGVTHIGIBJMT
|
6.3 | IC50 | 5 | — | |
HHSVICUMCOBRPT
|
6.3 | Ki | 33 | — |