Target Details
| UniProt AC | Q9H2X6 |
|---|---|
| Gene Symbol | HIPK2 |
| Protein Name | Homeodomain-interacting protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 256
- Clinical molecules 15
- Avg pChEMBL 6.86
KEGG Pathways (1)
Active Molecules (256)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KUNZDWIFPOMUOX
|
7.0 | Ki | 36 | — | |
MLDQJTXFUGDVEO
|
7.0 | IC50 | 85 | Yes | |
OBZHLULOFFWAJX
|
7.0 | Ki | 8 | — | |
PNKALLUVKOKYHZ
|
7.0 | Ki | 32 | — | |
SKKRZILJUKYLJS
|
7.0 | Ki | 25 | — | |
VVEGARMQKNYDID
|
7.0 | Ki | 24 | — | |
WLDOAHGSNVRGSC
|
7.0 | Ki | 4 | — | |
ZAOAKWGRHJIYTD
|
7.0 | Ki | 8 | — | |
NVTNPVQFMSQPJQ
|
7.0 | IC50 | 7 | — | |
OYONTEXKYJZFHA
|
7.0 | IC50 | 69 | Yes | |
OOLXXVMFVSTNLJ
|
6.9 | IC50 | 4 | — | |
ZCBUQCWBWNUWSU
|
6.9 | IC50 | 59 | — | |
KTGZHJWTKLQHBK
|
6.9 | IC50 | 3 | — | |
CHTMRWQLNNRRFJ
|
6.9 | Ki | 70 | — | |
DKSNLQYRZJKYOC
|
6.9 | Ki | 51 | — | |
DQPYZHUAILXFJI
|
6.9 | Ki | 27 | — | |
GCYXEGSPUDSZJY
|
6.9 | Ki | 82 | — | |
HKSZLNNOFSGOKW
|
6.9 | Ki | 118 | — | |
HOYRWTWZUFFACV
|
6.9 | Ki | 28 | — | |
HSMUWLLZAZCLHF
|
6.9 | Ki | 25 | — | |
LCHCSKHPVCDXAU
|
6.9 | Ki | 30 | — | |
RKDYDLMULRETNX
|
6.9 | Ki | 8 | — | |
RYAVJHIPOWNWDE
|
6.9 | Ki | 38 | — | |
UZFPGFONVYFSRR
|
6.9 | Ki | 16 | — | |
XOOAAYRIVATZNM
|
6.9 | Ki | 55 | — | |
XSRHBCYNCKAFKS
|
6.9 | Ki | 45 | — | |
BLQYVHBZHAISJM
|
6.8 | Ki | 54 | — | |
LACOMQAWPSFXQC
|
6.8 | Ki | 27 | — | |
LOMGAGWJYPGDLT
|
6.8 | Ki | 8 | — | |
LVECPYVAIBNSRV
|
6.8 | Ki | 33 | — | |
OQNPAZRZCXFOBC
|
6.8 | Ki | 11 | — | |
RVSKJUNTDGBSSS
|
6.8 | Ki | 25 | — | |
SMRWVXLSRJWVBF
|
6.8 | Ki | 25 | — | |
SQXSMLLCDWJNAC
|
6.8 | Ki | 20 | — | |
UFMAIBLTWQRHAK
|
6.8 | Ki | 10 | — | |
UXUQVXDYXKMCGA
|
6.8 | Ki | 21 | — | |
UYGYYOIUVFMGKQ
|
6.8 | Ki | 30 | — | |
WPHKIQPVPYJNAX
|
6.8 | Ki | 81 | — | |
WZISGNDZZPSYRP
|
6.8 | Ki | 20 | — | |
XJSFDMGICAWQFS
|
6.8 | Ki | 60 | — | |
LDNVJIDFNXGSGT
|
6.8 | IC50 | 6 | — | |
YEFYCSKFDBXSSK
|
6.8 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
6.7 | IC50 | 408 | — | |
DJUSDFVEBBYFFL
|
6.7 | Ki | 27 | — | |
DKXHSOUZPMHNIZ
|
6.7 | Ki | 51 | Yes | |
HNZBELVVHGZHII
|
6.7 | Ki | 5 | — | |
KRIUNPBAQZGFQA
|
6.7 | Ki | 76 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
NBLFGELIWIKRAC
|
6.7 | Ki | 8 | — | |
NHHQJBCNYHBUSI
|
6.7 | Ki | 220 | — |