Target Details
| UniProt AC | Q9H2K8 |
|---|---|
| Gene Symbol | TAOK3 |
| Protein Name | Serine/threonine-protein kinase TAO3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 73
- Clinical molecules 14
- Avg pChEMBL 7.0
KEGG Pathways (2)
Active Molecules (73)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
MPVGZUGXCQEXTM
|
6.6 | Kd | 61 | Yes | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
NXSJMRCTGYTSTK
|
6.4 | Kd | 200 | — | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
YRDHKIFCGOZTGD
|
6.4 | IC50 | 21 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
MFAQYJIYDMLAIM
|
6.3 | Kd | 130 | Yes | |
CTALVCVKEYVQIJ
|
6.3 | IC50 | 2 | — | |
KYAGDWQXJICEFO
|
6.3 | IC50 | 2 | — | |
MKUQVFUKAUXYEW
|
6.3 | IC50 | 2 | — | |
UBIKJGRVXIINFB
|
6.3 | IC50 | 2 | — | |
UKZSZOYTVQHXML
|
6.3 | IC50 | 2 | — | |
ZEGLWOVBWQUGAL
|
6.3 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.2 | Kd | 65 | — | |
OUSFTKFNBAZUKL
|
6.2 | Kd | 58 | Yes | |
YABJJWZLRMPFSI
|
6.1 | Kd | 34 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — |