Target Details
| UniProt AC | Q9H2K8 |
|---|---|
| Gene Symbol | TAOK3 |
| Protein Name | Serine/threonine-protein kinase TAO3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 73
- Clinical molecules 14
- Avg pChEMBL 7.0
KEGG Pathways (2)
Active Molecules (73)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
ODPGGGTTYSGTGO
|
8.2 | Kd | 153 | — | |
DKZYXHCYPUVGAF
|
7.7 | Kd | 112 | — | |
OYONTEXKYJZFHA
|
7.4 | Kd | 69 | Yes | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
CUIHSIWYWATEQL
|
7.3 | Kd | 61 | Yes | |
DGLFSNZWRYADFC
|
7.3 | IC50 | 12 | — | |
AJLWHEZEVCJFTK
|
7.3 | IC50 | 2 | — | |
BLXRLDWQFVTLLB
|
7.3 | IC50 | 2 | — | |
BMIWGAPTSPJEJO
|
7.3 | IC50 | 2 | — | |
BVNBRKOALNETGX
|
7.3 | IC50 | 2 | — | |
CHEWOUMVNNRPQL
|
7.3 | IC50 | 2 | — | |
CMHKKTGCFWZUEZ
|
7.3 | IC50 | 2 | — | |
CTTLBTOARINAOQ
|
7.3 | IC50 | 2 | — | |
CVJUGGSXRCYDMH
|
7.3 | IC50 | 2 | — | |
FEWKYLIQAFEHAS
|
7.3 | IC50 | 2 | — | |
FKLPOUDFRUNULX
|
7.3 | IC50 | 2 | — | |
HWNWXVSQBFOHFT
|
7.3 | IC50 | 2 | — | |
IWFBETHWIWFHFI
|
7.3 | IC50 | 2 | — | |
JRVGQZOVEXJARK
|
7.3 | IC50 | 2 | — | |
JSGUDZBCODXIII
|
7.3 | IC50 | 2 | — | |
JZZXFSWUEYNLNZ
|
7.3 | IC50 | 2 | — | |
LYJAJWGXMOKLOA
|
7.3 | IC50 | 2 | — | |
MBGWYGHZHAXUFZ
|
7.3 | IC50 | 2 | — | |
MJXKBVJFXOMGJZ
|
7.3 | IC50 | 2 | — | |
MLHQXLYJVYMVNC
|
7.3 | IC50 | 2 | — | |
MLYQDOZQEYXGTC
|
7.3 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.3 | Kd | 1075 | — | |
NWRZXVYYHQMCAU
|
7.3 | IC50 | 2 | — | |
OIEFVAVADRALOZ
|
7.3 | IC50 | 2 | — | |
OZYLOBCEPYGHNK
|
7.3 | IC50 | 2 | — | |
QLJIETHEHOPBEV
|
7.3 | IC50 | 2 | — | |
QLWPBOYRMFPURQ
|
7.3 | IC50 | 2 | — | |
QSAYKRXJXDKAIM
|
7.3 | IC50 | 2 | — | |
QTLUCZVJQWOZNL
|
7.3 | IC50 | 2 | — | |
SEJNBCOCDTVEAV
|
7.3 | IC50 | 2 | — | |
USKFTJSEVSYZHZ
|
7.3 | IC50 | 2 | — | |
UXGKCQZWBHGMBU
|
7.3 | IC50 | 2 | — | |
VCKRURAVBSHCHK
|
7.3 | IC50 | 2 | — | |
YBMXZSWZDVESLG
|
7.3 | IC50 | 2 | — | |
ZAGFGDPXBTWJKY
|
7.3 | IC50 | 2 | — | |
ZKPHMJAXPXACLF
|
7.3 | IC50 | 2 | — | |
ZZSRKSMPHPUYRC
|
7.3 | IC50 | 2 | — | |
OVPNQJVDAFNBDN
|
7.2 | Kd | 44 | Yes | |
GCIKSSRWRFVXBI
|
7.1 | Kd | 109 | Yes | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
ZCBUQCWBWNUWSU
|
7.0 | Kd | 59 | — | |
BIIVYFLTOXDAOV
|
7.0 | Kd | 82 | Yes | |
LCBAQTCTQXHTJG
|
6.9 | IC50 | 9 | — | |
JRNJNYBQQYBCLE
|
6.7 | Kd | 40 | Yes |